SCHEMBL7532041

SCHEMBL7532041

Fc1ccc(Cc2cccc(-c3n[nH]c4ccc(-c5ncn[nH]5)cc34)c2)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CLK2 P49760 3/20 0.52
DYRK1A Q13627 3/20 0.52
DYRK3 O43781 2/20 0.52
JAK2 O60674 2/20 0.52
PRKD3 O94806 2/20 0.52
MAP4K4 O95819 2/20 0.52
GSK3B P49841 2/20 0.52
JAK3 P52333 2/20 0.52
CSNK1G2 P78368 2/20 0.52
MELK Q14680 2/20 0.52
PRKD2 Q9BZL6 2/20 0.52
CLK4 Q9HAZ1 2/20 0.52
CSNK1G1 Q9HCP0 2/20 0.52
CSNK1G3 Q9Y6M4 2/20 0.52
GAK O14976 1/20 0.52
NQO2 P16083 1/20 0.52
CSNK2A2 P19784 1/20 0.52
FECH P22830 1/20 0.52
JAK1 P23458 1/20 0.52
TYK2 P29597 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL599945 0.84 MAP3K5 (0.50) CLK2DYRK1ADYRK3JAK2PRKD3
SCHEMBL5378711 0.81 MAPK8 (0.54) CLK2DYRK1ADYRK3JAK2PRKD3
SCHEMBL5375066 0.81 MAP3K5 (0.47) CLK2DYRK1ADYRK3JAK2PRKD3
SCHEMBL8252245 0.80 MAP3K5 (0.56) CLK2DYRK1ADYRK3JAK2PRKD3
SCHEMBL8365703 0.78 MKNK1 (0.60) CLK2DYRK1ADYRK3JAK2PRKD3
SCHEMBL5382298 0.77 GAK (0.56) CLK2DYRK1ADYRK3JAK2PRKD3
SCHEMBL5372315 0.77 IDO1 (0.69) CLK2DYRK1ADYRK3JAK2PRKD3
SCHEMBL8257010 0.77 ENPP2 (0.69) CLK2DYRK1ADYRK3JAK2PRKD3
SCHEMBL5381716 0.76 MAP3K5 (0.54) CLK2DYRK1ADYRK3JAK2PRKD3
SCHEMBL5375071 0.75 MAP3K5 (0.51) CLK2DYRK1ADYRK3JAK2PRKD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20020103229-A1 Indazole derivatives as JNK inhibitors and compositions and methods related thereto SIGNAL PHARMACEUTICALS, LLC 2002-08-01 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020103229-A1 Indazole derivatives as JNK inhibitors and compositions and methods related thereto MAP3K7, MAP3K1, MAP3K8 CLK2 322/4885DYRK1A 784/4885DYRK3 805/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.