SCHEMBL7532097

SCHEMBL7532097

N=C(N)N(CCOCCN(C(=N)N)C(=O)c1nc(Cl)c(N)nc1N)C(=O)c1nc(Cl)c(N)nc1N

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SCNN1A P37088 11/20 0.42
ALDH1A1 P00352 7/20 0.42
GLA P06280 6/20 0.42
HSD17B10 Q99714 6/20 0.42
KDM4E B2RXH2 5/20 0.42
HPGD P15428 5/20 0.42
GAA P10253 4/20 0.42
CYP1A2 P05177 4/20 0.42
PLAU P00749 3/20 0.42
SLC9A5 Q14940 3/20 0.42
CYP2D6 P10635 3/20 0.42
LMNA P02545 2/20 0.42
FTO Q9C0B1 2/20 0.42
BLM P54132 2/20 0.42
TSHR P16473 2/20 0.42
SLC22A1 O15245 1/20 0.42
HTR1A P08908 1/20 0.42
SLC9A1 P19634 1/20 0.42
MAOA P21397 1/20 0.42
ADORA2A P29274 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bromide SCHEMBL4693743 0.99 SCNN1A (0.41) SCNN1AALDH1A1GLAHSD17B10KDM4E
SCHEMBL7527745 0.99 SCNN1A (0.41) SCNN1AALDH1A1GLAHSD17B10KDM4E
Hydrochloric Acid SCHEMBL4751466 0.97 ALDH1A1 (0.43) SCNN1AALDH1A1GLAHSD17B10KDM4E
SCHEMBL4413401 0.94 SCNN1A (0.38) SCNN1AALDH1A1GLAHSD17B10KDM4E
Hydrochloric Acid SCHEMBL6013438 0.89 ALDH1A1 (0.36) SCNN1AALDH1A1GLAHSD17B10KDM4E
Hydrochloric Acid SCHEMBL4417773 0.87 KDM4E (0.39) SCNN1AALDH1A1GLAHSD17B10KDM4E
Bromide SCHEMBL4693421 0.86 SCNN1A (0.44) SCNN1AALDH1A1GLAHSD17B10KDM4E
Hydrochloric Acid SCHEMBL4693835 0.85 KDM4E (0.46) SCNN1AALDH1A1GLAHSD17B10KDM4E
Bromide SCHEMBL4789642 0.85 SCNN1A (0.43) SCNN1AALDH1A1GLAHSD17B10KDM4E
Hydrochloric Acid SCHEMBL6013436 0.84 KDM4E (0.38) SCNN1AALDH1A1GLAHSD17B10KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20020158255-A1 Conjugates of sodium channel blockers and methods of using the same NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2002-10-31 US disclosed