SCHEMBL7533643

SCHEMBL7533643

CCC(=O)c1ccc(C(N)=O)cc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.57
L3MBTL1 Q9Y468 2/20 0.57
SMN1; SMN2 Q16637 2/20 0.57
PARP10 Q53GL7 6/20 0.55
PARP4 Q9UKK3 2/20 0.50
PARP1 P09874 2/20 0.50
CA2 P00918 2/20 0.50
CA1 P00915 1/20 0.50
PARP2 Q9UGN5 1/20 0.50
ALDH1A1 P00352 2/20 0.48
KMT2A Q03164 1/20 0.48
PARP15 Q460N3 1/20 0.48
PARP14 Q460N5 1/20 0.48
PARP16 Q8N5Y8 1/20 0.48
PARP11 Q9NR21 1/20 0.48
TSHR P16473 2/20 0.48
POLB P06746 1/20 0.48
CYP3A4 P08684 1/20 0.48
CYP2C19 P33261 1/20 0.48
RECQL P46063 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8051337 0.87 SMN1; SMN2 (0.70) MAPTL3MBTL1SMN1; SMN2ALDH1A1KMT2A
Ethyne SCHEMBL8050785 0.82 SMN1; SMN2 (0.64) MAPTL3MBTL1SMN1; SMN2ALDH1A1KMT2A
SCHEMBL2677861 0.82 HSD17B3 (0.67) L3MBTL1SMN1; SMN2PARP10PARP4PARP1
SCHEMBL221282 0.81 MAPT (0.57) MAPTL3MBTL1SMN1; SMN2ALDH1A1KMT2A
SCHEMBL10389933 0.80 SMN1; SMN2 (0.83) MAPTL3MBTL1SMN1; SMN2ALDH1A1KMT2A
Terephthalamide SCHEMBL23774 0.79 PARP1 (0.71) MAPTL3MBTL1SMN1; SMN2PARP10PARP4
SCHEMBL31042968 0.79 CA2 (0.55) MAPTL3MBTL1SMN1; SMN2CA2ALDH1A1
SCHEMBL9448618 0.79 PARP1 (0.57) MAPTL3MBTL1SMN1; SMN2PARP10PARP1
SCHEMBL8282094 0.78 MAPT (0.59) MAPTL3MBTL1SMN1; SMN2ALDH1A1KMT2A
SCHEMBL2644065 0.78 SMN1; SMN2 (0.59) MAPTL3MBTL1SMN1; SMN2ALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002028353-A2 PHOSPHATE TRANSPORT INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2002-04-11 WO claimed
US-20100256755-A1 Poly(Tetrafluoroethene) Polymer With Nitric Oxide Donating Surface MEDTRONIC VASCULAR, INC. (US) 2010-10-07 US disclosed
WO-2002028353-A2 PHOSPHATE TRANSPORT INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2002-04-11 WO disclosed
CN-1336919-A Phenylphenanthridines with PDE-IV inhibiting activity BYK GULDEN LOMBERG CHEM FAB (DE) 2002-02-20 CN disclosed