SCHEMBL7538308

SCHEMBL7538308

CCN(C(=O)c1c(O)c2c(OC)cccc2n(C)c1=O)c1ccc(F)cc1F

nearest known ligand 0.54

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HDAC4 P56524 1/20 0.54
TP53 P04637 3/20 0.42
RORC P51449 1/20 0.40
TSHR P16473 2/20 0.39
BRPF1 P55201 1/20 0.38
HIF1A Q16665 4/20 0.37
CREBBP Q92793 2/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
MAPT P10636 3/20 0.36
THRB P10828 1/20 0.36
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
POLB P06746 2/20 0.36
PABPC1 P11940 1/20 0.36
LMNA P02545 1/20 0.35
GLA P06280 1/20 0.35
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7537746 0.93 HDAC4 (0.54) HDAC4TP53RORCTSHRBRPF1
SCHEMBL5163474 0.87 HDAC4 (0.64) HDAC4TP53RORCTSHRBRPF1
SCHEMBL7535425 0.86 HDAC4 (0.62) HDAC4TSHRMAPTMEN1KMT2A
SCHEMBL8151209 0.86 HDAC4 (0.39) HDAC4TP53TSHRHIF1AMEN1
SCHEMBL7620493 0.86 HDAC4 (0.39) HDAC4TP53TSHRHIF1ATHRB
SCHEMBL8151208 0.85 HDAC4 (0.38) HDAC4TP53TSHRHIF1AMAPT
SCHEMBL5165770 0.82 HDAC4 (0.59) HDAC4TP53TSHRBRPF1HIF1A
SCHEMBL5163897 0.82 HDAC4 (0.64) HDAC4TP53RORCTSHRBRPF1
SCHEMBL7533271 0.80 HDAC4 (0.40) HDAC4TP53RORCTSHRHIF1A
SCHEMBL6999887 0.79 HDAC4 (0.78) HDAC4RORCTSHRMAPTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20020173520-A1 Quinoline derivatives ACTIVE BIOTECH AB (SE) 2002-11-21 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020173520-A1 Quinoline derivatives CYP4F3, IRF3, CXCR3 HDAC4 2957/4885TP53 2677/4885RORC 603/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.