SCHEMBL7539558

SCHEMBL7539558

COc1cccc(-c2nnn[nH]2)c1C(=O)NCCCC(NC(=O)c1c(Cl)cccc1Cl)C(=O)O

nearest known ligand 0.44

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ITGA4 P13612 14/20 0.44
ITGB1 P05556 13/20 0.44
ITGB7 P26010 10/20 0.44
ITGA5 P08648 2/20 0.40
TAAR1 Q96RJ0 1/20 0.37
ITGB2 P05107 2/20 0.36
ICAM1 P05362 2/20 0.36
ITGAL P20701 2/20 0.36
ITGAV P06756 2/20 0.36
ITGB6 P18564 2/20 0.36
ITGB8 P26012 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7588676 0.85 ITGB1 (0.41) ITGA4ITGB1ITGB7ITGA5ITGB2
SCHEMBL7542115 0.85 TAAR1 (0.50) ITGA4ITGB1ITGB7ITGA5TAAR1
SCHEMBL7541262 0.82 TAAR1 (0.49) ITGA4ITGB1ITGB7ITGA5TAAR1
SCHEMBL7540693 0.82 TAAR1 (0.49) ITGA4ITGB1ITGB7ITGA5TAAR1
SCHEMBL7547311 0.80 HDAC3 (0.42) ITGA4ITGB1ITGB7ITGA5TAAR1
SCHEMBL7548629 0.78 ITGB1 (0.55) ITGA4ITGB1ITGB7ITGA5ITGB2
SCHEMBL7542016 0.77 TAS1R3 (0.50) ITGA4ITGB1ITGB7ITGA5TAAR1
SCHEMBL7539479 0.74 ITGB1 (0.54) ITGA4ITGB1ITGA5ITGB2ICAM1
SCHEMBL7540665 0.74 TAS1R3 (0.49) ITGA4ITGB1ITGB7ITGA5TAAR1
SCHEMBL7546250 0.74 TAS1R3 (0.49) ITGA4ITGB1ITGB7ITGA5TAAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1209147-A1 CARBOXYLIC ACID DERIVATIVES AND ADHESION MOLECULE INHIBITORS CONTAINING THE SAME AS THE ACTIVE INGREDIENT TORAY INDUSTRIES, INC. (JP) 2002-05-29 EP disclosed