SCHEMBL7540187

SCHEMBL7540187

COc1ccc(Br)c2c1C=C([N+](=O)[O-])CC2

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.47
CYP1A2 P05177 1/20 0.37
ALDH1A1 P00352 4/20 0.35
TDP1 Q9NUW8 3/20 0.35
HPGD P15428 2/20 0.34
GLA P06280 1/20 0.34
GAA P10253 1/20 0.34
POLB P06746 2/20 0.34
L3MBTL1 Q9Y468 2/20 0.34
CTDSP1 Q9GZU7 1/20 0.34
KMT2A Q03164 4/20 0.33
MEN1 O00255 3/20 0.33
MAPT P10636 2/20 0.33
MCOLN3 Q8TDD5 1/20 0.33
HTT P42858 1/20 0.33
AMY1A P0DUB6 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32
CYP19A1 P11511 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7547973 0.82 HTR2A (0.39) KDM4EALDH1A1MAPTHTTPTGS2
SCHEMBL7540781 0.81 MAPK1 (0.38) KDM4ECYP1A2ALDH1A1TDP1HPGD
SCHEMBL7543629 0.80 KMT2A (0.37) KDM4EALDH1A1TDP1HPGDGLA
SCHEMBL7543632 0.80 TDP1 (0.33) KDM4ECYP1A2ALDH1A1TDP1HPGD
SCHEMBL7546763 0.78 GRIN2D (0.36) KDM4EALDH1A1POLBKMT2AMEN1
Nitrous Acid SCHEMBL7549271 0.77 HTR2A (0.36) KDM4EMAPTHTTPTGS2
SCHEMBL30439274 0.68 TDP1 (0.51) KDM4EALDH1A1TDP1POLBL3MBTL1
SCHEMBL2494137 0.68 TDP1 (0.51) KDM4EALDH1A1TDP1POLBL3MBTL1
SCHEMBL25280185 0.67 TDP1 (0.51) KDM4EALDH1A1TDP1POLBL3MBTL1
SCHEMBL14142210 0.67 KDM4E (0.44) KDM4ECYP1A2ALDH1A1TDP1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0883599-B1 AMINOTETRALIN DERIVATIVES AND COMPOSITIONS AND METHOD OF USE THEREOF ASTRAZENECA AB (SE) 2002-06-05 EP disclosed
US-5807897-A MUSCULAR DISORDERS ZENECA LIMITED (GB) 1998-09-15 US disclosed