SCHEMBL7543632

SCHEMBL7543632

COc1ccc(CS)c2c1C=C([N+](=O)[O-])CC2

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 3/20 0.33
ALDH1A1 P00352 4/20 0.33
KDM4E B2RXH2 4/20 0.32
L3MBTL1 Q9Y468 3/20 0.32
POLB P06746 1/20 0.32
CTDSP1 Q9GZU7 1/20 0.32
GAA P10253 2/20 0.32
HPGD P15428 2/20 0.32
GLA P06280 1/20 0.32
MEN1 O00255 2/20 0.31
KMT2A Q03164 2/20 0.31
MAPT P10636 2/20 0.31
MAPK1 P28482 1/20 0.31
HTT P42858 2/20 0.31
CYP3A4 P08684 2/20 0.30
CYP2C9 P11712 2/20 0.30
CYP2C19 P33261 2/20 0.30
CYP19A1 P11511 1/20 0.30
PTGS2 P35354 1/20 0.30
CYP1A2 P05177 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7540781 0.80 MAPK1 (0.38) TDP1ALDH1A1KDM4EPOLBGAA
SCHEMBL7540187 0.80 KDM4E (0.47) TDP1ALDH1A1KDM4EL3MBTL1POLB
SCHEMBL7543629 0.76 KMT2A (0.37) TDP1ALDH1A1KDM4EL3MBTL1POLB
SCHEMBL7547973 0.70 HTR2A (0.39) ALDH1A1KDM4EMAPTMAPK1HTT
SCHEMBL7546763 0.67 GRIN2D (0.36) ALDH1A1KDM4EPOLBMEN1KMT2A
Nitrous Acid SCHEMBL7549271 0.66 HTR2A (0.36) KDM4EMAPTHTTPTGS2
SCHEMBL4652150 0.65 TDP1 (0.58) TDP1ALDH1A1L3MBTL1POLBHPGD
Bromide SCHEMBL4650887 0.64 TDP1 (0.57) TDP1ALDH1A1L3MBTL1POLBHPGD
SCHEMBL7007492 0.61 ALDH1A1 (0.41) TDP1ALDH1A1KDM4EL3MBTL1GLA
SCHEMBL5763685 0.60 NR1H4 (0.49) TDP1ALDH1A1KDM4EL3MBTL1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0883599-B1 AMINOTETRALIN DERIVATIVES AND COMPOSITIONS AND METHOD OF USE THEREOF ASTRAZENECA AB (SE) 2002-06-05 EP disclosed
US-5807897-A MUSCULAR DISORDERS ZENECA LIMITED (GB) 1998-09-15 US disclosed