SCHEMBL7540765

SCHEMBL7540765

CCCCC(CC)n1cnc2c(Cl)nc(C)nc21

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CRHR1 P34998 6/20 0.37
CDK1 P06493 2/20 0.33
CDK5 Q00535 1/20 0.33
PIK3CA P42336 1/20 0.32
PIK3CB P42338 1/20 0.32
MTOR P42345 1/20 0.32
PIK3CG P48736 1/20 0.32
PIK3C3 Q8NEB9 1/20 0.32
ADA P00813 3/20 0.32
PDE2A O00408 2/20 0.32
PDE4A P27815 1/20 0.32
PDE4B Q07343 1/20 0.32
PDE4C Q08493 1/20 0.32
PDE4D Q08499 1/20 0.32
KDM4E B2RXH2 1/20 0.32
ALDH1A1 P00352 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP3A4 P08684 1/20 0.32
ALOX15 P16050 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7626686 0.86 CDK1 (0.34) CRHR1CDK1CDK5KDM4E
SCHEMBL7570558 0.82 CNR2 (0.38) CRHR1
SCHEMBL1742776 0.77 ADA (0.47) CDK1ADAPDE2APDE4APDE4B
SCHEMBL29782919 0.77 LMNA (0.38) CDK1CDK5KDM4E
SCHEMBL1741408 0.76 ADA (0.49) CDK1ADAPDE2APDE4APDE4B
SCHEMBL30148781 0.76 CDK1 (0.41) CDK1CDK5PIK3CAPIK3CBMTOR
SCHEMBL1913380 0.76 CDK1 (0.41) CDK1CDK5PIK3CAPIK3CBMTOR
SCHEMBL18546882 0.75 ADA (0.43) CDK1ADAPDE2APDE4APDE4B
SCHEMBL21755891 0.75 ADA (0.43) CDK1ADAPDE2APDE4APDE4B
SCHEMBL17615377 0.75 CDK2 (0.50) CDK1CDK5KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6448261-B1 CORTICOTROPIN RELEASING FACTOR ANTAGONISTS; TREATING ANXIETY, DEPRESSION, AND OTHER PSYCHIATRIC AND NEUROLOGICAL DISORDERS BRISTOL-MYERS SQUIBB PHARMA COMPANY 2002-09-10 US disclosed
EP-0935601-A4 ARYLAMINO FUSED PYRIDINES AND PYRIMIDINES DU PONT PHARM CO (US) 2002-08-07 EP disclosed
US-6107300-A CORTICOTROPIN RELEASING FACTOR ANTAGONIST; PSYCHOLOGICAL DISORDERS DUPONT PHARMACEUTICALS (US) 2000-08-22 US disclosed
EP-0935601-A2 ARYLAMINO FUSED PYRIDINES AND PYRIMIDINES Du Pont Pharmaceuticals Company (US) 1999-08-18 EP disclosed
WO-1997035539-A2 ARYLAMINO FUSED PYRIDINES AND PYRIMIDINES DU PONT PHARMACEUTICALS COMPANY (US) 1997-10-02 WO disclosed