SCHEMBL7542890

SCHEMBL7542890

CCCC(Cc1ccc(O)c(O)c1)c1ccc2ccccc2c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 3/20 0.50
ESR2 Q92731 1/20 0.50
CYP3A4 P08684 7/20 0.47
CYP2D6 P10635 7/20 0.47
SLC6A2 P23975 7/20 0.47
SLC6A3 Q01959 7/20 0.47
SLC6A4 P31645 6/20 0.47
KCNH2 Q12809 5/20 0.47
IGF1R P08069 3/20 0.45
INSR P06213 2/20 0.45
ALOX15 P16050 3/20 0.44
ALOX12 P18054 3/20 0.44
KDM4E B2RXH2 2/20 0.44
MEN1 O00255 2/20 0.44
ALDH1A1 P00352 2/20 0.44
TP53 P04637 2/20 0.44
HPGD P15428 2/20 0.44
MAPK1 P28482 2/20 0.44
RECQL P46063 2/20 0.44
KMT2A Q03164 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16550376 0.81 CYP2D6 (0.70) ESR1ESR2CYP3A4CYP2D6SLC6A2
SCHEMBL14995802 0.76 ESR1 (0.57) ESR1ESR2CYP3A4CYP2D6SLC6A2
SCHEMBL10584005 0.73 UGT2B7 (0.46) CYP3A4CYP2D6SLC6A2SLC6A3SLC6A4
SCHEMBL7502486 0.73 UGT2B7 (0.46) CYP3A4CYP2D6SLC6A2SLC6A3SLC6A4
SCHEMBL6571270 0.72 UGT2B7 (0.49) CYP3A4CYP2D6SLC6A2SLC6A3SLC6A4
SCHEMBL27548723 0.71 HTR2A (0.49) ESR1ESR2CYP3A4CYP2D6SLC6A2
SCHEMBL19425427 0.71 TDP1 (0.50) ESR1ESR2CYP3A4CYP2D6SLC6A3
SCHEMBL10583568 0.71 CYP2D6 (0.43) CYP3A4CYP2D6SLC6A2SLC6A3SLC6A4
SCHEMBL10583789 0.71 CYP2D6 (0.43) CYP3A4CYP2D6SLC6A2SLC6A3SLC6A4
SCHEMBL10580403 0.71 CYP2D6 (0.43) CYP3A4CYP2D6SLC6A2SLC6A3SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1119351-A2 USE OF CATECHOL DERIVATIVES AS PROTEINASE INHIBITORS Grünenthal GmbH (DE) 2001-08-01 EP claimed
WO-2000019989-A2 USE OF CATECHOL DERIVATIVES AS PROTEINASE INHIBITORS Grünenthal GmbH (DE) 2000-04-13 WO claimed