SCHEMBL7543923

SCHEMBL7543923

COc1cccc2c1C(Br)C2

nearest known ligand 0.47

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 1/20 0.47
DRD2 P14416 7/20 0.45
DRD3 P35462 5/20 0.45
HTR1A P08908 2/20 0.44
CHRM2 P08172 2/20 0.44
CHRM1 P11229 2/20 0.44
CHRM3 P20309 2/20 0.44
DRD4 P21917 4/20 0.43
CYP19A1 P11511 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22837453 0.80 HTR2A (0.47) HTR2ADRD2DRD3HTR1ACHRM2
SCHEMBL7542801 0.80 HTR2A (0.47) HTR2ADRD2DRD3HTR1ACHRM2
SCHEMBL5034348 0.76 HTR2A (0.48) HTR2ADRD2DRD3HTR1ACHRM2
SCHEMBL20478471 0.76 CHRM2 (0.45) HTR2ADRD2DRD3HTR1ACHRM2
SCHEMBL3163101 0.74 HTR2A (0.43) HTR2ADRD2DRD3HTR1ADRD4
SCHEMBL10321230 0.73 DRD2 (0.46) HTR2ADRD2DRD3HTR1A
SCHEMBL20478601 0.73 CA12 (0.46) HTR2AHTR1A
SCHEMBL10321232 0.73 DRD2 (0.46) HTR2ADRD2DRD3HTR1A
SCHEMBL22837450 0.71 CETP (0.46) HTR2ADRD2DRD3HTR1A
SCHEMBL9870482 0.70 ABCB1 (0.64) HTR2ADRD2DRD3HTR1ACHRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0940386-B1 Benzocyclobutan compounds, their process for preparation and pharmaceutical compositions containing them SERVIER LAB (FR) 2002-05-22 EP disclosed
US-6107345-A ANTIDEPRESSANT; PSYCHOLOGICAL DISORDERS ADIR ET COMPAGNIE (FR) 2000-08-22 US disclosed
EP-0940386-A1 Benzocyclobutan compounds, their process for preparation and pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 1999-09-08 EP disclosed