SCHEMBL7544180

SCHEMBL7544180

CCOc1ccc(Cc2cc(C3CCNCC3)n(CCF)n2)cc1

nearest known ligand 0.41

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 12/20 0.41
KCNH2 Q12809 1/20 0.40
CNR2 P34972 1/20 0.39
ADRA1A P35348 1/20 0.39
HRH1 P35367 1/20 0.39
HRH3 Q9Y5N1 1/20 0.39
GPR4 P46093 1/20 0.38
PLAT P00750 1/20 0.35
ACACB O00763 1/20 0.35
SRC P12931 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5764465 0.89 CCR5 (0.46) CCR5KCNH2CNR2GPR4
Hydrochloric Acid SCHEMBL5765862 0.88 CCR5 (0.46) CCR5KCNH2CNR2GPR4
SCHEMBL5764335 0.81 CCR5 (0.48) CCR5KCNH2GPR4
SCHEMBL5764647 0.80 CCR5 (0.50) CCR5KCNH2
SCHEMBL7493987 0.79 MAPT (0.49) CCR5KCNH2GPR4
SCHEMBL7224003 0.79 HRH1 (0.48) CCR5KCNH2HRH1HRH3
SCHEMBL5763292 0.79 PLAT (0.42) CCR5PLAT
SCHEMBL5761438 0.79 PLAT (0.46) CCR5PLAT
SCHEMBL5762566 0.78 CCR5 (0.50) CCR5HRH1PLAT
Hydrochloric Acid SCHEMBL7660201 0.78 PLAT (0.42) CCR5PLAT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1171122-A4 PYRROLIDINE MODULATORS OF CHEMOKINE RECEPTOR ACTIVITY MERCK & CO INC (US) 2002-05-29 EP disclosed
EP-1171122-A1 PYRROLIDINE MODULATORS OF CHEMOKINE RECEPTOR ACTIVITY Merck & Co., Inc. (US) 2002-01-16 EP disclosed
US-6248755-B1 ANTIINFLAMMATORY AGENTS; ANTIALLERGENS; AUTOIMMUNE DISEASES MERCK & CO., INC. 2001-06-19 US disclosed
WO-2000059502-A1 PYRROLIDINE MODULATORS OF CHEMOKINE RECEPTOR ACTIVITY MERCK & CO., INC. (US) 2000-10-12 WO disclosed