SCHEMBL7546016

SCHEMBL7546016

COCCOCCOc1cc(C(=O)O)ccc1N

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGER4 P35408 1/20 0.50
EP300 Q09472 2/20 0.46
POLB P06746 1/20 0.46
CASP6 P55212 1/20 0.46
TSHR P16473 2/20 0.46
CA12 O43570 1/20 0.45
CA1 P00915 1/20 0.45
CA2 P00918 1/20 0.45
CA4 P22748 1/20 0.45
CA6 P23280 1/20 0.45
CA7 P43166 1/20 0.45
TPMT P51580 1/20 0.45
CA9 Q16790 1/20 0.45
CA14 Q9ULX7 1/20 0.45
CYP1A2 P05177 1/20 0.43
CYP2D6 P10635 1/20 0.43
SLC6A2 P23975 1/20 0.43
SCN1A P35498 1/20 0.43
SLC6A3 Q01959 1/20 0.43
KCNH2 Q12809 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7611997 0.87 CYP1A2 (0.48) PTGER4TSHRCA12CA1CA2
SCHEMBL979369 0.83 POLB (0.46) PTGER4POLBCASP6TSHRCA12
SCHEMBL1345863 0.82 MAPT (0.51) PTGER4TSHRCA12CA1CA2
SCHEMBL1436418 0.82 POLB (0.64) POLBCASP6TSHRCA12CA1
SCHEMBL5925659 0.81 TSHR (0.62) TSHRCYP1A2CYP2D6SLC6A2SCN1A
SCHEMBL8085032 0.81 ALDH1A1 (0.62) TSHRCYP1A2CYP2D6SLC6A2SCN1A
SCHEMBL881352 0.80 ALDH1A1 (0.52) PTGER4POLBCASP6TSHRCA12
SCHEMBL25375627 0.80 EP300 (0.45) PTGER4EP300POLBCASP6TSHR
SCHEMBL25377590 0.79 TSHR (0.47) EP300POLBCASP6TSHRCA12
SCHEMBL25376165 0.79 PARP1 (0.49) EP300POLBCASP6TSHRCA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1124788-A4 BIS(HALOETHYL)AMINOBENZENE DERIVATIVES SHIONOGI BIORES CORP (US) 2002-11-06 EP disclosed
EP-1124788-A2 BIS(HALOETHYL)AMINOBENZENE DERIVATIVES Shionogi Bioresearch Corporation (US) 2001-08-22 EP disclosed
WO-2000024361-A2 BIS(HALOETHYL)AMINOBENZENE DERIVATIVES SHIONOGI BIORESEARCH CORP. (US) 2000-05-04 WO disclosed