SCHEMBL7546199

SCHEMBL7546199

C1=C(c2c[nH]c3ncccc23)CCN2CCCC12

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK11 Q15759 1/20 0.50
MAPK14 Q16539 1/20 0.50
HTR2A P28223 1/20 0.48
HTR2C P28335 1/20 0.48
HTR2B P41595 1/20 0.48
TMEM97 Q5BJF2 1/20 0.45
SIGMAR1 Q99720 1/20 0.45
CDC7 O00311 8/20 0.45
CCNT1 O60563 2/20 0.45
CCNA2 P20248 2/20 0.45
CDK2 P24941 2/20 0.45
CDK9 P50750 2/20 0.45
RET P07949 3/20 0.43
GSK3B P49841 2/20 0.42
HTR1A P08908 1/20 0.42
SLC6A4 P31645 1/20 0.42
PLK4 O00444 1/20 0.42
JAK2 O60674 1/20 0.42
CCNB2 O95067 1/20 0.42
MAP4K4 O95819 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7543009 0.81 MAPK11 (0.50) MAPK11MAPK14HTR2ACDK9GSK3B
SCHEMBL7567570 0.79 MAPK11 (0.55) MAPK11MAPK14HTR2ASIGMAR1CCNT1
SCHEMBL2063653 0.75 TMEM97 (0.47) HTR2AHTR2CHTR2BTMEM97SIGMAR1
SCHEMBL26773930 0.75 HTR2A (0.65) HTR2AHTR2CHTR2BCDC7CCNT1
SCHEMBL26773932 0.75 HTR2A (0.65) HTR2AHTR2CHTR2BCDC7CCNT1
SCHEMBL26773936 0.75 HTR2A (0.65) HTR2AHTR2CHTR2BCDC7CCNT1
SCHEMBL12422661 0.72 TMEM97 (0.53) HTR2AHTR2CHTR2BTMEM97SIGMAR1
SCHEMBL21714635 0.71 HTR2A (0.51) HTR2AHTR2CHTR2BTMEM97SIGMAR1
SCHEMBL5850081 0.70 MAPK11 (0.81) MAPK11MAPK14CDK2GSK3BCDK1
SCHEMBL13064304 0.70 TMEM97 (0.59) HTR2AHTR2CHTR2BTMEM97SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1204662-A1 AZAINDOLES HAVING SEROTONIN RECEPTOR AFFINITY NPS Allelix Corp. (CA) 2002-05-15 EP disclosed
WO-2001012629-A1 AZAINDOLES HAVING SEROTONIN RECEPTOR AFFINITY NPS ALLELIX CORP. (US) 2001-02-22 WO disclosed