SCHEMBL7546347

SCHEMBL7546347

O=C1CN(Cc2ccccc2)CCN(Cc2ccccc2)CC(=O)N(Cc2ccccc2)CCN1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
APP P05067 1/20 0.52
HRH3 Q9Y5N1 1/20 0.52
SIGMAR1 Q99720 2/20 0.50
MCHR1 Q99705 1/20 0.49
DDB1 Q16531 1/20 0.48
CRBN Q96SW2 1/20 0.48
L3MBTL1 Q9Y468 1/20 0.48
PRMT5 O14744 1/20 0.47
WDR77 Q9BQA1 1/20 0.47
CYP2C9 P11712 2/20 0.44
CYP2C19 P33261 2/20 0.44
EPHX2 P34913 1/20 0.44
MAPT P10636 1/20 0.44
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44
NPC1 O15118 1/20 0.44
RAB9A P51151 1/20 0.44
SLC2A1 P11166 1/20 0.43
GRM5 P41594 1/20 0.43
ALDH1A1 P00352 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28499086 0.95 SIGMAR1 (0.51) APPHRH3SIGMAR1MCHR1DDB1
SCHEMBL220097 0.89 SIGMAR1 (0.62) SIGMAR1DDB1CRBNL3MBTL1CYP2C9
SCHEMBL10841960 0.88 APP (0.62) APPHRH3SIGMAR1MCHR1L3MBTL1
Hydrochloric Acid SCHEMBL10843610 0.86 APP (0.61) APPHRH3SIGMAR1MCHR1L3MBTL1
SCHEMBL5704266 0.83 SIGMAR1 (0.54) HRH3SIGMAR1MCHR1DDB1CRBN
SCHEMBL28497387 0.82 MCHR1 (0.57) APPHRH3SIGMAR1MCHR1DDB1
SCHEMBL8024414 0.80 SIGMAR1 (0.58) SIGMAR1DDB1CRBNCYP2C9CYP2C19
SCHEMBL7265760 0.79 DDB1 (0.48) SIGMAR1DDB1CRBNL3MBTL1CYP2C9
SCHEMBL13083472 0.77 MCHR1 (0.56) APPHRH3SIGMAR1MCHR1L3MBTL1
SCHEMBL930649 0.77 MCHR1 (0.56) APPHRH3SIGMAR1MCHR1PRMT5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0815091-B1 POLYAZACYCLOALKANE COMPOUNDS NYCOMED IMAGING AS (NO) 2002-06-12 EP disclosed
EP-0815091-A1 POLYAZACYCLOALKANE COMPOUNDS NYCOMED IMAGING AS (NO) 1998-01-07 EP disclosed
US-5705637-A Polyazacycloalkane compounds NYCOMED IMAGING AS (NO) 1998-01-06 US disclosed
US-5677446-A Polyazacycloalkane compounds NYCOMED IMAGING AS (NO) 1997-10-14 US disclosed
US-5631368-A Polyazacycloalkane compounds NYCOMED IMAGING AS (NO) 1997-05-20 US disclosed
WO-1996028433-A1 POLYAZACYCLOALKANE COMPOUNDS NYCOMED IMAGING A.S (NO) 1996-09-19 WO disclosed