SCHEMBL7546803

SCHEMBL7546803

c1cncc(Cc2cc(C3CCNCC3)[nH]n2)c1

nearest known ligand 0.48

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MKNK1 Q9BUB5 5/20 0.48
MKNK2 Q9HBH9 5/20 0.48
CDK9 P50750 4/20 0.45
IGF1R P08069 1/20 0.45
CCNT1 O60563 2/20 0.44
DRD2 P14416 1/20 0.43
DRD4 P21917 1/20 0.43
GSK3B P49841 1/20 0.42
PLAT P00750 1/20 0.42
CHRM2 P08172 2/20 0.41
CHRM1 P11229 2/20 0.41
CHRNB2 P17787 2/20 0.41
CHRM3 P20309 2/20 0.41
CHRNA4 P43681 2/20 0.41
ROCK2 O75116 1/20 0.40
ROCK1 Q13464 1/20 0.40
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
POLB P06746 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL5763738 0.99 MKNK1 (0.47) MKNK1MKNK2CDK9IGF1RCCNT1
SCHEMBL5764334 0.85 MKNK1 (0.47) MKNK1MKNK2DRD2DRD4MEN1
Hydrochloric Acid SCHEMBL5765492 0.84 GABRA1 (0.46) MKNK1MKNK2DRD2DRD4MEN1
SCHEMBL5760970 0.77 MKNK1 (0.60) MKNK1MKNK2CDK9CCNT1PLAT
SCHEMBL5762028 0.77 MKNK1 (0.45) MKNK1MKNK2CDK9IGF1RDRD2
Trifluoroacetic Acid SCHEMBL7547215 0.76 CDK2 (0.45) MKNK1MKNK2CDK9MEN1KMT2A
Trifluoroacetic Acid SCHEMBL5763412 0.76 CDK2 (0.45) MKNK1MKNK2CDK9MEN1KMT2A
SCHEMBL5763716 0.75 MKNK1 (0.48) MKNK1MKNK2CDK9CCNT1DRD2
SCHEMBL5765218 0.75 MKNK1 (0.70) MKNK1MKNK2DRD2DRD4PLAT
SCHEMBL5762663 0.74 MEN1 (0.63) MKNK1MKNK2CDK9IGF1RPLAT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1192133-A1 N-CYCLOPENTYL MODULATORS OF CHEMOKINE RECEPTOR ACTIVITY Merck & Co., Inc. (US) 2002-04-03 EP disclosed
WO-2000076972-A1 N-CYCLOPENTYL MODULATORS OF CHEMOKINE RECEPTOR ACTIVITY MERCK & CO., INC. (US) 2000-12-21 WO disclosed