SCHEMBL7547375

SCHEMBL7547375

CC(C/C=C/c1ccc2c(c1)OCO2)N(C)C(=O)OC(C)(C)C

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.49
NPC1 O15118 2/20 0.49
RAB9A P51151 2/20 0.49
HPGD P15428 2/20 0.49
GABRA1 P14867 2/20 0.48
GABRB2 P47870 2/20 0.48
TRPM8 Q7Z2W7 3/20 0.46
ALDH1A1 P00352 4/20 0.46
PGR P06401 1/20 0.46
AR P10275 1/20 0.46
MAOA P21397 1/20 0.46
SLC6A2 P23975 1/20 0.46
PDE4A P27815 1/20 0.46
KDR P35968 1/20 0.46
SLC6A3 Q01959 1/20 0.46
EPHX2 P34913 1/20 0.44
TRPV1 Q8NER1 1/20 0.43
GAA P10253 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
SOAT1 P35610 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7547378 1.00 KDM4E (0.49) KDM4ENPC1RAB9AHPGDGABRA1
SCHEMBL7548337 0.82 AAK1 (0.32) KDM4ENPC1RAB9AHPGDGABRA1
SCHEMBL7547370 0.82 AAK1 (0.32) KDM4ENPC1RAB9AHPGDGABRA1
SCHEMBL7554007 0.80 GRIK1 (0.45)
SCHEMBL7547697 0.80 GRIK1 (0.45)
SCHEMBL7547700 0.80 GRIK1 (0.45)
SCHEMBL24883777 0.79 TAAR1 (0.49) HPGDALDH1A1SLC6A2SLC6A3GAA
SCHEMBL30169770 0.79 TAAR1 (0.49) HPGDALDH1A1SLC6A2SLC6A3GAA
SCHEMBL25132039 0.79 TAAR1 (0.49) HPGDALDH1A1SLC6A2SLC6A3GAA
SCHEMBL7549401 0.78 AAK1 (0.41) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1214288-A1 PHARMACEUTICAL COMPOSITIONS AND METHODS FOR USE Targacept Inc. (US) 2002-06-19 EP disclosed
US-6337351-B1 AROMATIC OLEFIN AMINES TARGACEPT, INC. 2002-01-08 US disclosed
WO-2001017943-A1 PHARMACEUTICAL COMPOSITIONS AND METHODS FOR USE TARGACEPT, INC. (US) 2001-03-15 WO disclosed