SCHEMBL7547440

SCHEMBL7547440

CCn1nc(Cc2ccc(OC(F)(F)F)cc2)cc1C1CCN(CC2CC(N(C)[C@H](CC(C)C)C(=O)O)CC2c2cccc(F)c2)CC1

nearest known ligand 0.71

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 20/20 0.71
DRD3 P35462 1/20 0.71
SLC6A3 Q01959 1/20 0.71
KCNH2 Q12809 4/20 0.71

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL5764824 0.99 CCR5 (0.70) CCR5DRD3SLC6A3KCNH2
SCHEMBL7549793 0.93 CCR5 (0.73) CCR5KCNH2
Hydrochloric Acid SCHEMBL5763948 0.93 CCR5 (0.72) CCR5DRD3SLC6A3KCNH2
SCHEMBL7543474 0.93 CCR5 (0.72) CCR5KCNH2
Hydrochloric Acid SCHEMBL5763944 0.93 CCR5 (0.72) CCR5KCNH2
SCHEMBL7545290 0.93 CCR5 (0.72) CCR5KCNH2
Hydrochloric Acid SCHEMBL5764680 0.92 CCR5 (0.76) CCR5KCNH2
Hydrochloric Acid SCHEMBL5762837 0.92 CCR5 (0.72) CCR5KCNH2
SCHEMBL7541681 0.92 CCR5 (0.84) CCR5DRD3SLC6A3KCNH2
Hydrochloric Acid SCHEMBL5765284 0.92 CCR5 (0.72) CCR5KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1192133-A1 N-CYCLOPENTYL MODULATORS OF CHEMOKINE RECEPTOR ACTIVITY Merck & Co., Inc. (US) 2002-04-03 EP disclosed
WO-2000076972-A1 N-CYCLOPENTYL MODULATORS OF CHEMOKINE RECEPTOR ACTIVITY MERCK & CO., INC. (US) 2000-12-21 WO disclosed