SCHEMBL7552013

SCHEMBL7552013

Cc1cc(COc2ccc(C(=O)NC3(C(C)C(=O)NO)CCOCC3)cc2)c2ccccc2n1.Cc1cc(COc2ccc(C(=O)NC3(CC(=O)NO)CCCCCC3)cc2)c2ccccc2n1

nearest known ligand 0.78

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ADAM17 P78536 19/20 0.78
ADAMTS4 O75173 2/20 0.78
MMP3 P08254 2/20 0.78
MMP7 P09237 2/20 0.78
ADAMTS1 Q9UHI8 2/20 0.78
ADAMTS5 Q9UNA0 2/20 0.78
MMP8 P22894 1/20 0.67
MMP13 P45452 1/20 0.63

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6597542 0.91 ADAM17 (0.71) ADAM17ADAMTS4MMP3MMP7ADAMTS1
SCHEMBL6599983 0.88 ADAM17 (1.00) ADAM17ADAMTS4MMP3MMP7ADAMTS1
SCHEMBL6597320 0.88 ADAM17 (1.00) ADAM17ADAMTS4MMP3MMP7ADAMTS1
SCHEMBL6597759 0.88 ADAM17 (1.00) ADAM17ADAMTS4MMP3MMP7ADAMTS1
SCHEMBL6595027 0.88 ADAM17 (0.98) ADAM17ADAMTS4MMP3MMP7ADAMTS1
Trifluoroacetic Acid SCHEMBL6597061 0.87 ADAM17 (0.66) ADAM17ADAMTS4MMP3MMP7ADAMTS1
SCHEMBL6597835 0.87 ADAM17 (0.67) ADAM17ADAMTS4MMP3MMP7ADAMTS1
SCHEMBL6600065 0.86 ADAM17 (0.95) ADAM17ADAMTS4MMP3MMP7ADAMTS1
SCHEMBL6594466 0.85 ADAM17 (0.83) ADAM17ADAMTS4MMP3MMP7ADAMTS1
SCHEMBL6595495 0.85 ADAM17 (0.83) ADAM17ADAMTS4MMP3MMP7ADAMTS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1263756-A2 BETA-AMINO ACID DERIVATIVES AS INHIBITORS OF MATRIX METALLOPROTEASES AND TNF-ALPHA Bristol-Myers Squibb Pharma Company (US) 2002-12-11 EP claimed
WO-2001070734-A2 BETA-AMINO ACID DERIVATIVES AS INHIBITORS OF MATRIX METALLOPROTEASES AND TNF-ALPHA BRISTOL-MYERS SQUIBB PHARMA COMPANY (US) 2001-09-27 WO claimed