SCHEMBL7555015

SCHEMBL7555015

CCOC(=O)N(C)c1c(C(=O)c2cnoc2C2CC2)ccc(Cl)c1Cl

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 3/20 0.35
KMT2A Q03164 3/20 0.33
SLC6A2 P23975 2/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
MEN1 O00255 2/20 0.33
RAB9A P51151 2/20 0.33
NPC1 O15118 1/20 0.33
MAPT P10636 2/20 0.33
POLB P06746 1/20 0.33
ALDH1A1 P00352 4/20 0.33
LMNA P02545 2/20 0.33
HPGD P15428 1/20 0.33
GPBAR1 Q8TDU6 1/20 0.32
MAPK1 P28482 2/20 0.32
HTT P42858 2/20 0.32
USP2 O75604 1/20 0.32
DHODH Q02127 3/20 0.32
SCN9A Q15858 1/20 0.32
SLC6A3 Q01959 1/20 0.31
PDE2A O00408 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7552560 0.89 SLC6A4 (0.35) SLC6A4KMT2ASLC6A2SMN1; SMN2MEN1
SCHEMBL7553925 0.89 DHODH (0.34) SLC6A4KMT2ASMN1; SMN2MEN1POLB
SCHEMBL7550436 0.86 SYK (0.35) SLC6A4KMT2AMEN1LMNAGPBAR1
SCHEMBL7552995 0.85 DHODH (0.34) SLC6A4KMT2AMEN1GPBAR1DHODH
SCHEMBL7552998 0.84 DHODH (0.36) SLC6A4KMT2AMEN1GPBAR1DHODH
SCHEMBL7643223 0.83 ALDH1A1 (0.36) KMT2ASMN1; SMN2MEN1RAB9ANPC1
SCHEMBL7550989 0.82 DHODH (0.33) SLC6A4KMT2ASLC6A2MEN1DHODH
SCHEMBL7551998 0.82 ALDH1A1 (0.31) SLC6A4SLC6A2SMN1; SMN2ALDH1A1
SCHEMBL8492602 0.82 CYP4F2 (0.36) SLC6A4SLC6A2MAPTALDH1A1LMNA
SCHEMBL7552797 0.81 DHODH (0.32) DHODH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0734380-B1 4-BENZOYLISOXAZOLES AND THEIR USE AS HERBICIDES AVENTIS AGRICULTURE LTD (GB) 2002-07-10 EP claimed
US-5658858-A POSTEMERGENCE HERBICIDES RHONE-POULENC ARGRICULTURE LIMITED (GB) 1997-08-19 US claimed
EP-0734380-A1 4-BENZOYLISOXAZOLES AND THEIR USE AS HERBICIDES RHONE-POULENC AGRICULTURE LTD. (GB) 1996-10-02 EP claimed
WO-1995016678-A1 4-BENZOYLISOXAZOLES AND THEIR USE AS HERBICIDES RHONE POULENC AGRICULTURE LIMITED (GB) 1995-06-22 WO claimed
EP-0734380-B1 4-BENZOYLISOXAZOLES AND THEIR USE AS HERBICIDES AVENTIS AGRICULTURE LTD (GB) 2002-07-10 EP disclosed
US-6369270-B1 CHEMICAL INTERMEDIATES RHONE POULENC AGRICULTURE LIMITED (GB) 2002-04-09 US disclosed
US-6114538-A 2-POSITION OF BENZOY RING OF 4-BENZOYLISOXAZOLE DERIVATIVE IS SUBSTITUTED AND PARTICULARLY USED AGAINST MONOCOTYLEDONOUS WEEDS BY POST-EMEREGENECE APPLICATION RHONE POULENC AGRICULTURE LIMITED (GB) 2000-09-05 US disclosed
US-5998653-A CHEMICAL INTERMEDIATE FOR HERBICIDES RHONE POULENC AGRICULTURE LIMITED (GB) 1999-12-07 US disclosed
US-5658858-A POSTEMERGENCE HERBICIDES RHONE-POULENC ARGRICULTURE LIMITED (GB) 1997-08-19 US disclosed
EP-0734380-A1 4-BENZOYLISOXAZOLES AND THEIR USE AS HERBICIDES RHONE-POULENC AGRICULTURE LTD. (GB) 1996-10-02 EP disclosed
WO-1995022903-A1 NEW PESTICIDAL METHOD RHONE-POULENC AGROCHIMIE (FR) 1995-08-31 WO disclosed
WO-1995016678-A1 4-BENZOYLISOXAZOLES AND THEIR USE AS HERBICIDES RHONE POULENC AGRICULTURE LIMITED (GB) 1995-06-22 WO disclosed