SCHEMBL7555058

SCHEMBL7555058

COc1ccc2c(ccn2-c2ccccc2C#N)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK1 Q13464 1/20 0.45
PTK2 Q05397 1/20 0.44
L3MBTL1 Q9Y468 5/20 0.44
POLB P06746 2/20 0.44
HTR6 P50406 1/20 0.44
PDGFRB P09619 1/20 0.44
PDGFRA P16234 1/20 0.44
GAA P10253 1/20 0.42
MEN1 O00255 3/20 0.41
MAPT P10636 3/20 0.41
KMT2A Q03164 3/20 0.41
KDM4E B2RXH2 3/20 0.41
NCOA1 Q15788 2/20 0.41
NCOA3 Q9Y6Q9 2/20 0.41
HTT P42858 2/20 0.41
MAPK1 P28482 2/20 0.41
TDP1 Q9NUW8 2/20 0.41
LMNA P02545 1/20 0.41
PABPC1 P11940 1/20 0.41
CASP3 P42574 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28037181 0.82 MAOB (0.43) ROCK1PTK2GAAMAPTKMT2A
SCHEMBL6660146 0.79 HSP90AA1 (0.43) ROCK1PTK2KMT2AKDM4ELMNA
SCHEMBL31116815 0.79 ROCK1 (0.51) ROCK1L3MBTL1POLBHTR6PDGFRB
SCHEMBL28842817 0.79 ROCK1 (0.48) ROCK1L3MBTL1POLBHTR6PDGFRB
SCHEMBL1270502 0.79 MAT2A (0.44) PTK2GAAMEN1KMT2AKDM4E
SCHEMBL31454935 0.79 ROCK1 (0.54) ROCK1L3MBTL1POLBHTR6PDGFRB
SCHEMBL30097476 0.78 BIRC5 (0.43) ROCK1PTK2MEN1KMT2AKDM4E
SCHEMBL699112 0.78 BIRC5 (0.43) ROCK1PTK2MEN1KMT2AKDM4E
SCHEMBL16383852 0.76 KMT2A (0.43) PTK2L3MBTL1MEN1MAPTKMT2A
SCHEMBL4580723 0.75 ROCK1 (0.43) ROCK1L3MBTL1POLBHTR6PDGFRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1165512-A2 METHOD FOR ARYLATING AZA-HETEROCYCLES WITH ACTIVATED AROMATIC COMPOUNDS IN THE PRESENCE OF CESIUM CARBONATE GÖDECKE GMBH (DE) 2002-01-02 EP disclosed
WO-2000059883-A2 METHOD FOR PRODUCING N-ARYL-AZA-HETEROCYCLES IN THE PRESENCE OF CESIUM CARBONATE Gödecke GmbH (DE) 2000-10-12 WO disclosed