SCHEMBL7562437

SCHEMBL7562437

OC(Cn1ccnc1)c1ccc(F)cc1

nearest known ligand 0.72

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 3/20 0.72
HMOX1 P09601 1/20 0.67
CYP51A1 Q16850 1/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6299999 1.00 CYP19A1 (0.72) CYP19A1HMOX1CYP51A1
SCHEMBL10932073 0.85 CYP19A1 (0.73) CYP19A1HMOX1CYP51A1
SCHEMBL11633201 0.84 CYP19A1 (0.73) CYP19A1HMOX1
SCHEMBL11983140 0.84 CYP19A1 (0.72) CYP19A1HMOX1CYP51A1
SCHEMBL4313095 0.84 CYP19A1 (0.72) CYP19A1HMOX1CYP51A1
SCHEMBL11266884 0.84 CYP19A1 (0.72) CYP19A1HMOX1CYP51A1
SCHEMBL10197408 0.84 HMOX1 (0.91) CYP19A1HMOX1CYP51A1
SCHEMBL10816487 0.84 HMOX1 (0.91) CYP19A1HMOX1CYP51A1
SCHEMBL6173273 0.83 CYP19A1 (0.71) CYP19A1HMOX1CYP51A1
SCHEMBL6299346 0.83 CYP19A1 (0.71) CYP19A1HMOX1CYP51A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 14 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115894461-B Novel coumarin-containing azole derivative, and preparation method and application thereof 沈阳药科大学 2024-01-23 CN disclosed
CN-115028585-B Arylalkylazole derivative and application thereof 聊城大学 2023-08-18 CN disclosed
CN-115894461-A Novel coumarin azole-containing derivative and preparation method and application thereof 沈阳药科大学 2023-04-04 CN disclosed
CN-115028585-A Arylalkanazole derivatives and use thereof 聊城大学 2022-09-09 CN disclosed
CN-109320458-B Diaryl imidazole-containing compound, preparation method and medical application thereof 中国药科大学 2022-05-31 CN disclosed
CN-112694472-A BuChE-IDO1 inhibitor, preparation method and application thereof 西南大学 2021-04-23 CN disclosed
US-20020058665-A1 Imidazole derivatives and their use as farnesyl protein transferase inhibitors ASTRAZENECA UK LIMITED 2002-05-16 US disclosed
US-20020052376-A1 Imidazole derivatives and their use as farnesyl protein transferase inhibitors ASTRAZENECA UK LIMITED 2002-05-02 US disclosed
US-6342765-B1 COMPOUNDS THAT INHIBIT FARNESYLATION OF MUTANT RAS GENE PRODUCTS; TREATING DISEASES, ESPECIALLY CANCER, WHICH ARE MEDIATED THROUGH FARNESYLATION OF RAS ASTRAZENECA UK LIMITED (GB) 2002-01-29 US disclosed
EP-1025088-B1 IMIDAZOLE DERIVATIVES AND THEIR USE AS FARNESYL PROTEIN TRANSFERASE INHIBITORS ASTRAZENECA AB (SE) 2001-09-05 EP disclosed
EP-1025088-A1 IMIDAZOLE DERIVATIVES AND THEIR USE AS FARNESYL PROTEIN TRANSFERASE INHIBITORS AstraZeneca UK Limited (GB) 2000-08-09 EP disclosed
WO-1999020611-A1 IMIDAZOLE DERIVATIVES AND THEIR USE AS FARNESYL PROTEIN TRANSFERASE INHIBITORS ZENECA LIMITED (GB) 1999-04-29 WO disclosed
EP-0276583-A1 Imidazole derivatives, processes for their preparation and their fungicidal properties Instituto de Investigacion Y Desarrollo Quimico Biologico S.A. (ES) 1988-08-03 EP disclosed
US-4349556-A Pesticidally active 1-acyloxy-1-phenyl-2-azolyl-ethanes BAYER AKTIENGESELLSCHAFT (DE) 1982-09-14 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020058665-A1 Imidazole derivatives and their use as farnesyl protein transferase inhibitors FNTA, FNTB, RABGGTA CYP19A1 836/4885HMOX1 4023/4885CYP51A1 75/4885
US-20020052376-A1 Imidazole derivatives and their use as farnesyl protein transferase inhibitors FNTA, FNTB, RABGGTA CYP19A1 806/4885HMOX1 3930/4885CYP51A1 107/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.