SCHEMBL7562637

SCHEMBL7562637

COCc1c(-c2ccc(F)cc2)[c]c(C(C)C)nc1-c1ccccc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GCGR P47871 1/20 0.44
DPP4 P27487 1/20 0.37
HMGCR P04035 3/20 0.35
ESR1 P03372 1/20 0.35
CHRM1 P11229 1/20 0.35
TBXA2R P21731 1/20 0.35
PDE4A P27815 1/20 0.35
ADRA1A P35348 1/20 0.35
ADORA1 P30542 3/20 0.34
MAPK14 Q16539 1/20 0.33
ADORA2A P29274 1/20 0.33
SQOR Q9Y6N5 1/20 0.33
PTGDR2 Q9Y5Y4 2/20 0.33
SLC2A1 P11166 1/20 0.33
DHODH Q02127 1/20 0.33
SCN9A Q15858 1/20 0.33
HTR2A P28223 1/20 0.33
HTR2C P28335 1/20 0.33
HTR2B P41595 1/20 0.33
MEN1 O00255 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL526996 0.84 GCGR (0.56) GCGRHMGCRESR1CHRM1TBXA2R
SCHEMBL8846697 0.75 DHODH (0.40) GCGRDHODH
SCHEMBL9302519 0.72 ADORA2A (0.43) MAPK14ADORA2ASCN9AMEN1KMT2A
SCHEMBL7592397 0.68 ADORA2A (0.38) GCGRADORA1MAPK14ADORA2AHTR2A
SCHEMBL7559726 0.67 DPP4 (0.40) DPP4ADORA1ADORA2AHTR2AHTR2C
SCHEMBL7720729 0.66 GCGR (0.86) GCGRHMGCRESR1CHRM1TBXA2R
SCHEMBL8846284 0.66 MAPT (0.43) ADORA1ADORA2ASQORDHODHMEN1
SCHEMBL13115444 0.66 MAPK14 (0.53) GCGRMAPK14MEN1KMT2A
SCHEMBL9302391 0.64 APP (0.42) DHODHMEN1KMT2A
SCHEMBL8703691 0.64 ACP1 (0.41) ADORA2ADHODHMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0705837-B1 Preparation of 3-Oxy-5-oxo-6-heptenoic acid derivatives UBE INDUSTRIES (JP) 2002-08-07 EP disclosed
US-5744604-A Preparation of 3-oxy-5-oxo-6-heptenoic acid derivatives UBE INDUSTRIES, LTD. (JP) 1998-04-28 US disclosed
US-5677455-A Preparation of 3-oxy-5-oxo-6-heptenoic acid derivatives UBE INDUSTRIES, LTD. (JP) 1997-10-14 US disclosed
EP-0705837-A2 Preparation of 3-Oxy-5-oxo-6-heptenoic acid derivatives UBE INDUSTRIES, LTD. (JP) 1996-04-10 EP disclosed