SCHEMBL7565211

SCHEMBL7565211

CC1(C)C(=O)C(c2ccc(S(C)(=O)=O)cc2)=C1c1ccccc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 20/20 1.00
PTGS1 P23219 13/20 1.00
ABCB11 O95342 1/20 0.52
ALDH1A1 P00352 1/20 0.52
MT-CO2 P00403 1/20 0.52
HTR1A P08908 1/20 0.52
ADORA3 P0DMS8 1/20 0.52
MC4R P32245 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3832067 1.00 PTGS2 (1.00) PTGS2PTGS1ABCB11ALDH1A1MT-CO2
SCHEMBL7567995 0.94 PTGS2 (0.88) PTGS2PTGS1
SCHEMBL7565288 0.86 PTGS2 (1.00) PTGS2PTGS1
SCHEMBL7573838 0.86 PTGS2 (0.76) PTGS2PTGS1
SCHEMBL7567996 0.86 PTGS2 (1.00) PTGS2PTGS1
SCHEMBL7569451 0.86 PTGS2 (0.76) PTGS2PTGS1ABCB11ALDH1A1MT-CO2
SCHEMBL7567543 0.84 PTGS2 (0.72) PTGS2PTGS1ABCB11ALDH1A1MT-CO2
SCHEMBL7567551 0.84 PTGS2 (0.72) PTGS2PTGS1ABCB11ALDH1A1MT-CO2
SCHEMBL7568422 0.83 PTGS2 (0.73) PTGS2PTGS1
SCHEMBL7568223 0.83 PTGS2 (0.73) PTGS2PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0889878-B1 BISARYLCYCLOBUTENE DERIVATES AS CYCLOOXYGENASE INHIBITORS MERCK FROSST CANADA INC (CA) 2002-09-04 EP claimed
EP-0889878-B1 BISARYLCYCLOBUTENE DERIVATES AS CYCLOOXYGENASE INHIBITORS MERCK FROSST CANADA INC (CA) 2002-09-04 EP disclosed
WO-2002045704-A2 PREVENTION AND TREATMENT OF TACHYPHYLACTIC RESPONSE MOLECULAR SKINCARE LIMITED (GB) 2002-06-13 WO disclosed
EP-0889878-A1 BISARYLCYCLOBUTENE DERIVATES AS CYCLOOXYGENASE INHIBITORS MERCK FROSST CANADA INC. (CA) 1999-01-13 EP disclosed
US-5817700-A ANTIINFLAMMATORY AGENTS MERCK FROSST CANADA, INC. (CA) 1998-10-06 US disclosed
WO-1997036863-A1 BISARYLCYCLOBUTENE DERIVATES AS CYCLOOXYGENASE INHIBITORS MERCK FROSST CANADA INC. (CA) 1997-10-09 WO disclosed