SCHEMBL7567569

SCHEMBL7567569

CC(C)(C)C[C@H](NC(=O)N1CCOCC1)C(=O)N[C@H](C#N)CCc1ccccc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CTSS P25774 19/20 1.00
CTSL P07711 3/20 0.70
CTSB P07858 2/20 0.70

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6806938 0.90 CTSS (0.88) CTSSCTSLCTSB
SCHEMBL13937579 0.90 CTSS (0.82) CTSSCTSLCTSB
SCHEMBL6803089 0.88 CTSS (1.00) CTSSCTSLCTSB
SCHEMBL7062841 0.88 CTSS (1.00) CTSSCTSLCTSB
SCHEMBL7394849 0.87 CTSS (0.77) CTSSCTSLCTSB
SCHEMBL7543883 0.86 CTSS (1.00) CTSSCTSLCTSB
SCHEMBL7398906 0.86 CTSS (0.75) CTSSCTSLCTSB
SCHEMBL7395131 0.83 CTSS (0.83) CTSSCTSLCTSB
SCHEMBL6796532 0.83 CTSS (0.84) CTSSCTSLCTSB
SCHEMBL7391487 0.83 CTSS (0.88) CTSSCTSLCTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2002538151-A 2002-11-12 JP claimed
EP-1159273-A1 COMPOUNDS USEFUL AS REVERSIBLE INHIBITORS OF CATHEPSIN S BOEHRINGER INGELHEIM PHARMACEUTICALS INC. (US) 2001-12-05 EP claimed
WO-2000051998-A1 COMPOUNDS USEFUL AS REVERSIBLE INHIBITORS OF CATHEPSIN S BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 2000-09-08 WO claimed