SCHEMBL7567609

SCHEMBL7567609

CCCCc1ccc(S(=O)(=O)n2cc(C3=CCN(C)CC3)c3c(F)cccc32)cc1

nearest known ligand 0.58

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 17/20 0.58
DRD2 P14416 2/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C9 P11712 1/20 0.38
HTR2A P28223 1/20 0.38
HTR2C P28335 1/20 0.38
CYP2C19 P33261 1/20 0.38
DRD3 P35462 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4671200 0.84 HTR6 (0.61) HTR6CYP3A4CYP2D6
SCHEMBL3338517 0.77 HTR6 (0.51) HTR6
SCHEMBL4673875 0.74 HTR6 (1.00) HTR6CYP3A4CYP2D6
SCHEMBL4676436 0.71 HTR6 (1.00) HTR6DRD2CYP3A4CYP2D6
SCHEMBL4674305 0.70 HTR6 (0.82) HTR6CYP3A4CYP2D6
SCHEMBL7485051 0.69 HTR6 (0.79) HTR6
SCHEMBL4671281 0.69 HTR6 (0.76) HTR6CYP3A4CYP2D6
SCHEMBL4670653 0.68 HTR6 (0.80) HTR6
SCHEMBL3335540 0.68 HTR6 (0.80) HTR6DRD2CYP3A4CYP2D6
SCHEMBL4671653 0.67 HTR6 (0.76) HTR6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1173432-A1 PIPERIDINE-INDOLE COMPOUNDS HAVING 5-HT6 AFFINITY NPS Allelix Corp. (CA) 2002-01-23 EP disclosed
WO-2000063203-A1 PIPERIDINE-INDOLE COMPOUNDS HAVING 5-HT6 AFFINITY ALLELIX BIOPHARMACEUTICALS INC. (CA) 2000-10-26 WO disclosed