SCHEMBL7568665

SCHEMBL7568665

COC(=O)c1cccc(CON=C2C(c3ccccc3)=C(c3ccc(S(C)(=O)=O)cc3)C2(C)C)c1

nearest known ligand 0.48

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 8/20 0.48
PTGS1 P23219 5/20 0.47
ADAMTS4 O75173 1/20 0.42
MMP13 P45452 1/20 0.42
CA12 O43570 1/20 0.41
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
CA9 Q16790 1/20 0.41
MAPT P10636 1/20 0.40
MRGPRX4 Q96LA9 1/20 0.38
LOXL2 Q9Y4K0 1/20 0.38
CYP4F2 P78329 1/20 0.37
CYP4A11 Q02928 1/20 0.37
ACLY P53396 1/20 0.37
CD74 P04233 1/20 0.37
MIF P14174 1/20 0.37
PLAU P00749 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7573854 0.92 PTGS2 (0.49) PTGS2PTGS1ADAMTS4MMP13CA1
SCHEMBL7570401 0.86 PTGS2 (0.60) PTGS2PTGS1
SCHEMBL7568518 0.86 PTGS2 (0.60) PTGS2PTGS1
SCHEMBL7568513 0.86 PTGS2 (0.60) PTGS2PTGS1
SCHEMBL7570406 0.86 PTGS2 (0.60) PTGS2PTGS1
SCHEMBL7568732 0.79 PTGS2 (0.51) PTGS2PTGS1
SCHEMBL7568735 0.79 PTGS2 (0.51) PTGS2PTGS1
SCHEMBL7567226 0.76 PTGS2 (0.67) PTGS2PTGS1
SCHEMBL7567230 0.76 PTGS2 (0.67) PTGS2PTGS1
SCHEMBL7569113 0.74 PTGS2 (0.53) PTGS2PTGS1ADAMTS4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0889878-B1 BISARYLCYCLOBUTENE DERIVATES AS CYCLOOXYGENASE INHIBITORS MERCK FROSST CANADA INC (CA) 2002-09-04 EP claimed