SCHEMBL7569592

SCHEMBL7569592

NCCc1ccccc1Br.NCCc1ccccc1C(F)(F)F

nearest known ligand 0.69

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 8/20 0.69
MAOB P27338 2/20 0.49
IDO1 P14902 3/20 0.47
DAO P14920 1/20 0.43
HDAC1 Q13547 1/20 0.40
HDAC8 Q9BY41 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
CA5A P35218 1/20 0.39
CA9 Q16790 1/20 0.39
HTR2A P28223 1/20 0.38
HTR2C P28335 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29915506 0.89 MAOB (0.57) TAAR1MAOBIDO1DAOHDAC1
SCHEMBL1011004 0.89 MAOB (0.57) TAAR1MAOBIDO1DAOHDAC1
Iodide SCHEMBL28682742 0.87 MAOB (0.55) TAAR1MAOBIDO1DAOHDAC1
Hydrochloric Acid SCHEMBL6944674 0.87 MAOB (0.59) TAAR1MAOBIDO1DAOSMN1; SMN2
SCHEMBL29423333 0.83 TAAR1 (1.00) TAAR1IDO1SMN1; SMN2HTR2AHTR2C
SCHEMBL265615 0.83 TAAR1 (1.00) TAAR1IDO1SMN1; SMN2HTR2AHTR2C
Bromide SCHEMBL31622102 0.81 TAAR1 (0.95) TAAR1IDO1SMN1; SMN2HTR2AHTR2C
Iodide SCHEMBL28685278 0.81 TAAR1 (0.95) TAAR1IDO1SMN1; SMN2HTR2AHTR2C
Hydrochloric Acid SCHEMBL533785 0.81 TAAR1 (0.95) TAAR1IDO1SMN1; SMN2HTR2AHTR2C
SCHEMBL2096671 0.78 IDO1 (0.53) TAAR1MAOBIDO1DAOHDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1144399-A3 HETEROCYCLIC CARBOXAMIDE-CONTAINING THIOUREA INHIBITORS OF HERPES VIRUSES CONTAINING A SUBSTITUTED PHENYLENEDIAMINE GROUP Wyeth (US) 2002-09-11 EP disclosed
EP-1144399-A2 HETEROCYCLIC CARBOXAMIDE-CONTAINING THIOUREA INHIBITORS OF HERPES VIRUSES CONTAINING A SUBSTITUTED PHENYLENEDIAMINE GROUP AMERICAN HOME PRODUCTS CORPORATION (US) 2001-10-17 EP disclosed
WO-2000034261-A2 HETEROCYCLIC CARBOXAMIDE-CONTAINING THIOUREA INHIBITORS OF HERPES VIRUSES CONTAINING A SUBSTITUTED PHENYLENEDIAMINE GROUP AMERICAN HOME PRODUCTS CORPORATION (US) 2000-06-15 WO disclosed