SCHEMBL7570569

SCHEMBL7570569

CCS(=O)(=O)N1CC2(CCN(C(=O)[C@@H](COCc3ccccc3)NC(=O)C(C)(C)N)CC2)c2ccccc21

nearest known ligand 0.87

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
GHSR Q92847 1/20 0.87
TACR1 P25103 19/20 0.65

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7570564 1.00 GHSR (0.87) GHSRTACR1
Hydrochloric Acid SCHEMBL7566530 0.99 GHSR (0.85) GHSRTACR1
Hydrochloric Acid SCHEMBL7566534 0.99 GHSR (0.85) GHSRTACR1
Ibutamoren SCHEMBL29369919 0.93 GHSR (1.00) GHSRTACR1
Ibutamoren SCHEMBL739398 0.93 GHSR (1.00) GHSRTACR1
Ibutamoren SCHEMBL4927761 0.93 GHSR (1.00) GHSRTACR1
Ibutamoren SCHEMBL4451194 0.92 GHSR (0.98) GHSRTACR1
Ibutamoren SCHEMBL7413830 0.92 GHSR (0.98) GHSRTACR1
Ibutamoren SCHEMBL7413834 0.92 GHSR (0.98) GHSRTACR1
Ibutamoren SCHEMBL29366896 0.92 GHSR (0.98) GHSRTACR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0615977-B1 Spiro piperidines and homologs which promote release of growth hormone MERCK & CO INC (US) 2002-07-03 EP disclosed
US-5652235-A Method of using spiro piperidines to promote the release of growth hormone MERCK & CO., INC. (US) 1997-07-29 US disclosed
US-5536716-A Spiro piperidines and homologs which promote release of growth hormone MERCK & CO., INC. (US) 1996-07-16 US disclosed
EP-0615977-A1 Spiro piperidines and homologs which promote release of growth hormone MERCK & CO. INC. (US) 1994-09-21 EP disclosed