SCHEMBL7570925

SCHEMBL7570925

CCCCC/C=C\C/C=C\CCCCCCCC(=O)C(OP(=O)(O)OCCN)(C(=O)CCCCCCC/C=C\C/C=C\CCCCC)[C@@H](O)CO

nearest known ligand 0.48

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 1/20 0.47
SELP P16109 1/20 0.46
ALDH1A1 P00352 1/20 0.45
MAPT P10636 1/20 0.45
THRB P10828 1/20 0.45
CNR1 P21554 1/20 0.45
KDM4E B2RXH2 2/20 0.43
SOAT1 P35610 1/20 0.43
P2RY10 O00398 4/20 0.42
GPR34 Q9UPC5 1/20 0.42
FABP3 P05413 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5312425 0.97 ALDH1A1 (0.48) S1PR1SELPALDH1A1MAPTTHRB
SCHEMBL969822 0.97 P2RY10 (0.44) S1PR1P2RY10GPR34
SCHEMBL18262003 0.97 P2RY10 (0.44) S1PR1P2RY10GPR34
SCHEMBL7571747 0.97 P2RY10 (0.44) S1PR1P2RY10GPR34
SCHEMBL7573946 0.94 FABP3 (0.42) S1PR1SELPALDH1A1MAPTTHRB
SCHEMBL19410782 0.91 PLA2G2C (0.43) P2RY10GPR34
SCHEMBL37519 0.91 PLA2G2C (0.43) P2RY10GPR34
SCHEMBL226745 0.91 PLA2G2C (0.43) P2RY10GPR34
SCHEMBL3963403 0.91 PLA2G2C (0.43) P2RY10GPR34
SCHEMBL17144721 0.91 PLA2G2C (0.43) P2RY10GPR34

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0845981-B1 COMPOSITIONS COMPRISING CATIONIC AMPHIPHILES AND CO-LIPIDS FOR INTRACELLULAR DELIVERY OF THERAPEUTIC MOLECULES GENZYME CORP (US) 2002-09-25 EP claimed
US-5935936-A A DRUG DELIVERY FOR GENE THERAPY COMPRISING A DIAMINO-POLY-ALKYLAMINE-CARBAMOYL CHOLESTEROL AND AT LEAST ONE PHOSPHATIDES GENZYME CORPORATION (US) 1999-08-10 US claimed
EP-0845981-A1 COMPOSITIONS COMPRISING CATIONIC AMPHIPHILES AND CO-LIPIDS FOR INTRACELLULAR DELIVERY OF THERAPEUTIC MOLECULES GENZYME CORPORATION (US) 1998-06-10 EP claimed
WO-1997046223-A1 COMPOSITIONS COMPRISING CATIONIC AMPHIPHILES AND CO-LIPIDS FOR INTRACELLULAR DELIVERY OF THERAPEUTIC MOLECULES GENZYME CORPORATION (US) 1997-12-11 WO claimed
EP-4337179-A1 METHODS FOR TREATING, AMELIORATING OR PREVENTING INFECTIONS USING DRUG AND VACCINATION COMBINATION TREATMENT Topelia Aust Limited (ACN 652 771 670) (AU) 2024-03-20 EP disclosed
WO-2024006937-A1 LIPID COMPOSITIONS FOR IN VIVO DELIVERY Life Technologies Corporation (US) 2024-01-04 WO disclosed
WO-2023092060-A1 MICRORNA-DEPENDENT MRNA SWITCHES FOR TISSUE-SPECIFIC MRNA-BASED THERAPIES CORNELL UNIVERSITY (US) 2023-05-25 WO disclosed
WO-2021222304-A1 SARS-COV-2 RNA VACCINES MODERNATX, INC. (US) 2021-11-04 WO disclosed
EP-0845981-B1 COMPOSITIONS COMPRISING CATIONIC AMPHIPHILES AND CO-LIPIDS FOR INTRACELLULAR DELIVERY OF THERAPEUTIC MOLECULES GENZYME CORP (US) 2002-09-25 EP disclosed
US-5935936-A A DRUG DELIVERY FOR GENE THERAPY COMPRISING A DIAMINO-POLY-ALKYLAMINE-CARBAMOYL CHOLESTEROL AND AT LEAST ONE PHOSPHATIDES GENZYME CORPORATION (US) 1999-08-10 US disclosed
EP-0845981-A1 COMPOSITIONS COMPRISING CATIONIC AMPHIPHILES AND CO-LIPIDS FOR INTRACELLULAR DELIVERY OF THERAPEUTIC MOLECULES GENZYME CORPORATION (US) 1998-06-10 EP disclosed
WO-1997046223-A1 COMPOSITIONS COMPRISING CATIONIC AMPHIPHILES AND CO-LIPIDS FOR INTRACELLULAR DELIVERY OF THERAPEUTIC MOLECULES GENZYME CORPORATION (US) 1997-12-11 WO disclosed