SCHEMBL7571215

SCHEMBL7571215

CN(c1nccc(-n2cnc3ccccc32)n1)C1CCN(C(=O)OCc2ccccc2)CC1

nearest known ligand 0.60

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
LCK P06239 7/20 0.60
GRIN2B Q13224 5/20 0.44
SMN1; SMN2 Q16637 3/20 0.44
NPC1 O15118 2/20 0.44
RAB9A P51151 2/20 0.44
GPR119 Q8TDV5 1/20 0.44
CYP2C19 P33261 1/20 0.43
IDH1 O75874 1/20 0.43
MKNK2 Q9HBH9 2/20 0.43
MKNK1 Q9BUB5 1/20 0.43
CYP2D6 P10635 1/20 0.42
CYP2C9 P11712 1/20 0.42
FAAH O00519 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7505588 0.95 LCK (0.62) LCKGRIN2BSMN1; SMN2NPC1RAB9A
SCHEMBL7506273 0.90 LCK (0.67) LCKMKNK2MKNK1
SCHEMBL7990480 0.84 LCK (0.60) LCKGRIN2BSMN1; SMN2NPC1RAB9A
SCHEMBL7502002 0.83 LCK (0.66) LCKIDH1MKNK2MKNK1
SCHEMBL7505777 0.80 LCK (0.82) LCKGRIN2BCYP2D6CYP2C9
SCHEMBL7547581 0.80 LCK (0.53) LCKGPR119
SCHEMBL7570454 0.78 LCK (0.62) LCKMKNK2MKNK1
SCHEMBL7508722 0.77 LCK (0.91) LCKGRIN2BCYP2D6CYP2C9
SCHEMBL7547951 0.76 LCK (0.57) LCK
SCHEMBL7986459 0.76 LCK (0.52) LCKMKNK2MKNK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1206260-A4 SRC KINASE INHIBITOR COMPOUNDS MERCK & CO INC (US) 2002-10-30 EP disclosed
EP-1206260-A1 SRC KINASE INHIBITOR COMPOUNDS Merck & Co., Inc. (US) 2002-05-22 EP disclosed
WO-2001000207-A1 SRC KINASE INHIBITOR COMPOUNDS MERCK & CO., INC. (US) 2001-01-04 WO disclosed