SCHEMBL757175

SCHEMBL757175

O=c1c2c(F)cccc2nc(CSc2ncnc3[nH]ncc23)n1Cc1ccccc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CG P48736 8/20 0.49
PIK3CD O00329 4/20 0.42
MET P08581 1/20 0.41
ALDH1A1 P00352 3/20 0.41
ALDH1A2 O94788 1/20 0.41
ALDH1A3 P47895 1/20 0.41
HSD17B10 Q99714 1/20 0.41
RXFP1 Q9HBX9 1/20 0.41
PIK3R1 P27986 1/20 0.40
POLB P06746 2/20 0.40
RECQL P46063 1/20 0.40
PIK3CA P42336 1/20 0.40
PIK3CB P42338 1/20 0.40
HPGD P15428 1/20 0.40
TP53 P04637 1/20 0.39
MAPT P10636 1/20 0.39
HTT P42858 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
GAA P10253 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL734521 0.83 PIK3CG (0.55) PIK3CGPIK3CDALDH1A1HSD17B10RXFP1
SCHEMBL17805206 0.79 PIK3CG (0.47) PIK3CGPIK3CDALDH1A1HSD17B10RXFP1
SCHEMBL18548675 0.76 PIK3CG (0.51) PIK3CGPIK3CDALDH1A1HSD17B10RXFP1
SCHEMBL732945 0.75 PIK3CG (0.69) PIK3CGPIK3CDALDH1A1HSD17B10RXFP1
SCHEMBL10296666 0.73 LMNA (0.56) PIK3CGPIK3CDALDH1A1HSD17B10RXFP1
SCHEMBL734970 0.72 PIK3CG (0.52) PIK3CGPIK3CDALDH1A1HSD17B10RXFP1
SCHEMBL732815 0.71 PIK3CG (0.51) PIK3CGPIK3CDALDH1A1HSD17B10RXFP1
SCHEMBL18526831 0.69 PIK3CD (0.46) PIK3CGPIK3CDHSD17B10PIK3R1PIK3CA
SCHEMBL734922 0.68 PIK3CD (0.60) PIK3CGPIK3CDHSD17B10PIK3R1PIK3CA
SCHEMBL735026 0.68 PIK3CG (0.77) PIK3CGPIK3CDALDH1A1HSD17B10RXFP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8138195-B2 Inhibitors of human phosphatidylinositol 3-kinase delta ICOS CORPORATION (US) 2012-03-20 US disclosed
US-8138195-B2 Inhibitors of human phosphatidylinositol 3-kinase delta ICOS CORPORATION (US) 2012-03-20 US disclosed