SCHEMBL7572356

SCHEMBL7572356

CCOC(=O)C[C@@H](CC(C)C)N(Cc1ccccc1)[C@H](C)c1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.42
HSD17B10 Q99714 2/20 0.42
LMNA P02545 2/20 0.42
POLB P06746 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
F10 P00742 1/20 0.42
F2 P00734 1/20 0.42
TSHR P16473 1/20 0.41
TP53 P04637 2/20 0.40
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
CHRNB2 P17787 1/20 0.38
CHRNB4 P30926 1/20 0.38
CHRNA3 P32297 1/20 0.38
CHRNA4 P43681 1/20 0.38
ALOX5 P09917 2/20 0.37
PPID Q08752 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
MAPT P10636 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4196740 0.91 ALDH1A1 (0.41) ALDH1A1HSD17B10LMNAPOLBL3MBTL1
SCHEMBL4196745 0.91 ALDH1A1 (0.41) ALDH1A1HSD17B10LMNAPOLBL3MBTL1
SCHEMBL4192209 0.90 ALDH1A1 (0.40) ALDH1A1HSD17B10LMNAPOLBL3MBTL1
SCHEMBL5188655 0.90 ALDH1A1 (0.40) ALDH1A1HSD17B10LMNAPOLBL3MBTL1
SCHEMBL4192216 0.90 ALDH1A1 (0.40) ALDH1A1HSD17B10LMNAPOLBL3MBTL1
SCHEMBL2311421 0.89 ALDH1A1 (0.43) ALDH1A1HSD17B10LMNAPOLBL3MBTL1
SCHEMBL2311414 0.89 ALDH1A1 (0.43) ALDH1A1HSD17B10LMNAPOLBL3MBTL1
SCHEMBL4208000 0.88 F10 (0.39) ALDH1A1HSD17B10LMNAPOLBL3MBTL1
SCHEMBL4207996 0.88 F10 (0.39) ALDH1A1HSD17B10LMNAPOLBL3MBTL1
SCHEMBL14231825 0.87 ALDH1A1 (0.41) ALDH1A1HSD17B10LMNAPOLBL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6114328-A ANTICOAGULANTS; BLOOD DISORDERS DUPONT PHARMACEUTICALS COMPANY (US) 2000-09-05 US disclosed
EP-0970950-A2 Novel isoxazoline and isoxazole fibrinogen receptor antagonists DuPont Pharmaceuticals Company (US) 2000-01-12 EP disclosed
US-5849736-A Isoxazoline and isoxazole fibrinogen receptor antagonists THE DUPONT MERCK PHARMACEUTICAL COMPANY (US) 1998-12-15 US disclosed
WO-1995014683-A1 NOVEL ISOXAZOLINE AND ISOXAZOLE FIBRINOGEN RECEPTOR ANTAGONISTS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1995-06-01 WO disclosed