SCHEMBL7573300

SCHEMBL7573300

CNC(=O)c1nccnc1OC

nearest known ligand 0.41

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MAPT P10636 1/20 0.41
TSHR P16473 1/20 0.41
PLK1 P53350 2/20 0.40
KDM4E B2RXH2 1/20 0.36
HPGDS O60760 2/20 0.36
SMN1; SMN2 Q16637 2/20 0.35
YTHDC1 Q96MU7 1/20 0.34
PRKCI P41743 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
ALDH1A1 P00352 3/20 0.34
NPC1 O15118 1/20 0.34
TP53 P04637 1/20 0.34
PKM P14618 1/20 0.34
RAB9A P51151 1/20 0.34
GRM4 Q14833 1/20 0.34
GAA P10253 1/20 0.34
IRAK4 Q9NWZ3 1/20 0.34
HPGD P15428 1/20 0.33
TYK2 P29597 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24993555 0.83 P2RX7 (0.42) MAPTTSHRKDM4ESMN1; SMN2PRKCI
SCHEMBL31140247 0.83 P2RX7 (0.42) MAPTTSHRKDM4ESMN1; SMN2PRKCI
SCHEMBL31214279 0.80 NPSR1 (0.48) MAPTTSHRKDM4EL3MBTL1ALDH1A1
SCHEMBL958881 0.80 NPSR1 (0.48) MAPTTSHRKDM4EL3MBTL1ALDH1A1
SCHEMBL31172397 0.79 SCD (0.38) MAPTTSHRSMN1; SMN2YTHDC1L3MBTL1
SCHEMBL30592770 0.78 MAPT (0.47) MAPTTSHRKDM4EL3MBTL1ALDH1A1
SCHEMBL336307 0.78 BCHE (0.39) MAPTTSHRKDM4ESMN1; SMN2L3MBTL1
SCHEMBL1111686 0.78 MAPT (0.47) MAPTTSHRKDM4EL3MBTL1ALDH1A1
SCHEMBL17674836 0.76 MAPT (0.36) MAPTTSHRKDM4ESMN1; SMN2L3MBTL1
SCHEMBL2215923 0.76 CDC7 (0.46) MAPTTSHRPLK1KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1196384-A4 1-(AROMATIC- OR HETEROAROMATIC-SUBSTITUTED)-3-(HETEROAROMATIC SUBSTITUTED)-1,3-PROPANEDIONES AND USES THEREOF MERCK & CO INC (US) 2002-10-23 EP disclosed
EP-1196384-A1 1-(AROMATIC- OR HETEROAROMATIC-SUBSTITUTED)-3-(HETEROAROMATIC SUBSTITUTED)-1,3-PROPANEDIONES AND USES THEREOF Merck & Co., Inc. (US) 2002-04-17 EP disclosed
WO-2001000578-A1 1-(AROMATIC- OR HETEROAROMATIC-SUBSTITUTED)-3-(HETEROAROMATIC SUBSTITUTED)-1,3-PROPANEDIONES AND USES THEREOF MERCK & CO., INC. (US) 2001-01-04 WO disclosed