SCHEMBL7573372

SCHEMBL7573372

Clc1cccc(C#CC/N=C/c2ccccc2)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM5 P08912 1/20 0.41
CYP2D6 P10635 2/20 0.40
KCNH2 Q12809 1/20 0.39
GRIN1 Q05586 4/20 0.38
GRIN2B Q13224 4/20 0.38
LMNA P02545 1/20 0.38
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
GRM5 P41594 2/20 0.36
CYP2C9 P11712 1/20 0.36
PTGDR2 Q9Y5Y4 1/20 0.36
CHRM2 P08172 1/20 0.36
CHRM1 P11229 1/20 0.36
GRIN2D O15399 2/20 0.35
GRIN3B O60391 2/20 0.35
GRIN2A Q12879 2/20 0.35
GRIN2C Q14957 2/20 0.35
GRIN3A Q8TCU5 2/20 0.35
PTGES O14684 1/20 0.34
MMP13 P45452 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7573374 1.00 CHRM5 (0.41) CHRM5CYP2D6KCNH2GRIN1GRIN2B
SCHEMBL7571671 0.93 CHRM5 (0.50) CHRM5CYP2D6KCNH2GRIN1GRIN2B
SCHEMBL7571676 0.93 CHRM5 (0.50) CHRM5CYP2D6KCNH2GRIN1GRIN2B
SCHEMBL7574454 0.91 CYP2D6 (0.40) CHRM5CYP2D6KCNH2GRIN1GRIN2B
SCHEMBL7574457 0.91 CYP2D6 (0.40) CHRM5CYP2D6KCNH2GRIN1GRIN2B
SCHEMBL7578987 0.91 CHRM5 (0.49) CHRM5CYP2D6GRIN1GRIN2BLMNA
SCHEMBL7578981 0.91 CHRM5 (0.49) CHRM5CYP2D6GRIN1GRIN2BLMNA
SCHEMBL7571250 0.84 CYP1A2 (0.45) LMNACYP2C9MEN1CYP1A2MAPT
SCHEMBL7571246 0.84 CYP1A2 (0.45) LMNACYP2C9MEN1CYP1A2MAPT
SCHEMBL7579055 0.83 G6PC1 (0.43) GRIN1GRIN2BLMNANPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0810199-B1 Method for producing propargylamine compounds SUMITOMO CHEMICAL CO (JP) 2002-09-25 EP disclosed
US-5756769-A Method for producing propargylamine compounds SUMITOMO CHEMICAL COMPANY, LTD. (JP) 1998-05-26 US disclosed
EP-0810199-A1 Method for producing propargylamine compounds SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1997-12-03 EP disclosed