SCHEMBL7573709

SCHEMBL7573709

COc1cccc(Oc2c(NS(=O)(=O)c3ccc(C)cc3S)cc(C(=O)O)cc2OCC(O)CO)c1

nearest known ligand 0.46

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
EDNRB P24530 1/20 0.46
TSHR P16473 1/20 0.40
MAPK1 P28482 1/20 0.40
FABP4 P15090 3/20 0.38
MRGPRX1 Q96LB2 1/20 0.36
SLC16A3 O15427 2/20 0.36
ALDH1A1 P00352 2/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
RAD52 P43351 1/20 0.35
PTGDR2 Q9Y5Y4 2/20 0.34
CPT2 P23786 1/20 0.34
CPT1A P50416 1/20 0.34
ACLY P53396 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7568104 0.92 EDNRB (0.57) EDNRBTSHRMAPK1ALDH1A1SMN1; SMN2
SCHEMBL7570801 0.89 EDNRB (0.42) EDNRBTSHRMAPK1ALDH1A1ACLY
SCHEMBL7566571 0.85 EDNRB (0.56) EDNRBTSHRMAPK1SLC16A3ALDH1A1
SCHEMBL7567636 0.83 EDNRB (0.52) EDNRB
SCHEMBL7567507 0.81 EDNRB (0.66) EDNRBTSHRMAPK1SLC16A3ALDH1A1
SCHEMBL7569419 0.78 EDNRB (0.54) EDNRBTSHRMAPK1ALDH1A1SMN1; SMN2
SCHEMBL7569202 0.78 EDNRB (0.70) EDNRBALDH1A1SMN1; SMN2MEN1KMT2A
SCHEMBL7565566 0.77 EDNRB (0.51) EDNRB
SCHEMBL8771691 0.77 EDNRB (0.49) EDNRBMAPK1ALDH1A1SMN1; SMN2MEN1
SCHEMBL7568255 0.76 EDNRB (0.65) EDNRBALDH1A1SMN1; SMN2MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0799206-B1 ARYL- AND HETARYL-SULFONAMIDE DERIVATIVES, THEIR PREPARATION AND THEIR USE AS ENDOTHELIN ANTAGONISTS HOFFMANN LA ROCHE (CH) 2002-09-11 EP claimed