SCHEMBL7574431

SCHEMBL7574431

C#C/C(N)=C\c1ccc(C)cc1C

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.40
KMT2A Q03164 3/20 0.40
TDP1 Q9NUW8 3/20 0.36
SLC9A3 P48764 2/20 0.36
TP53 P04637 1/20 0.36
SLC9A1 P19634 1/20 0.36
GABRA1 P14867 1/20 0.36
GABRG2 P18507 1/20 0.36
GABRB3 P28472 1/20 0.36
AMY1A P0DUB6 1/20 0.36
CYP1A1 P04798 1/20 0.33
CYP1B1 Q16678 1/20 0.33
MAPT P10636 4/20 0.33
LMNA P02545 3/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
KDM4E B2RXH2 1/20 0.33
POLB P06746 1/20 0.33
HSP90AA1 P07900 1/20 0.33
ALOX12 P18054 1/20 0.33
HTT P42858 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8261303 0.79 TDP1 (0.43) MEN1KMT2ATDP1SLC9A3TP53
SCHEMBL7581821 0.78 ALDH1A1 (0.42) MEN1KMT2ATDP1TP53MAPT
SCHEMBL7579202 0.73 GRIN2D (0.41) TDP1MAPTLMNASMN1; SMN2KDM4E
SCHEMBL9550627 0.72 TDP1 (0.44) MEN1KMT2ATDP1SLC9A3TP53
SCHEMBL7572617 0.71 TP53 (0.46) MEN1KMT2ATDP1SLC9A3TP53
SCHEMBL1927493 0.70 KMT2A (0.58) MEN1KMT2ATDP1TP53GABRA1
SCHEMBL24496899 0.69 TDP1 (0.41) MEN1KMT2ATDP1SLC9A3TP53
SCHEMBL14402929 0.69 TDP1 (0.41) MEN1KMT2ATDP1SLC9A3TP53
SCHEMBL17225192 0.69 TDP1 (0.41) MEN1KMT2ATDP1SLC9A3TP53
SCHEMBL6392202 0.69 SLC9A3 (0.44) MEN1KMT2ATDP1SLC9A3TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0810199-B1 Method for producing propargylamine compounds SUMITOMO CHEMICAL CO (JP) 2002-09-25 EP disclosed
US-5756769-A Method for producing propargylamine compounds SUMITOMO CHEMICAL COMPANY, LTD. (JP) 1998-05-26 US disclosed
EP-0810199-A1 Method for producing propargylamine compounds SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1997-12-03 EP disclosed