SCHEMBL7576472

SCHEMBL7576472

O=C(O)C1=Nc2ccccc2C1=Cc1ccccc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLK1 P53350 1/20 0.43
MAPT P10636 6/20 0.42
KMT2A Q03164 6/20 0.42
MEN1 O00255 5/20 0.42
HPGD P15428 4/20 0.42
L3MBTL1 Q9Y468 3/20 0.42
TDP1 Q9NUW8 2/20 0.42
CDC25A P30304 1/20 0.42
CDC25B P30305 1/20 0.42
CTDSP1 Q9GZU7 1/20 0.42
KDM4E B2RXH2 5/20 0.41
PIM1 P11309 1/20 0.39
CYP19A1 P11511 1/20 0.37
CYP11B2 P19099 1/20 0.37
GSK3B P49841 1/20 0.36
LMNA P02545 3/20 0.36
ALDH1A1 P00352 3/20 0.36
POLB P06746 2/20 0.36
ALOX12 P18054 2/20 0.36
MCL1 Q07820 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27845629 0.75 PLK1 (0.41) PLK1MAPTKMT2AMEN1HPGD
SCHEMBL28698373 0.75 PLK1 (0.41) PLK1MAPTKMT2AMEN1HPGD
SCHEMBL27848261 0.73 MAPT (0.46) PLK1MAPTKMT2AMEN1HPGD
SCHEMBL6651141 0.72 MAPT (0.38) MAPTKMT2AMEN1HPGDL3MBTL1
SCHEMBL18229432 0.72 MAPT (0.45) MAPTKMT2AMEN1HPGDL3MBTL1
SCHEMBL5812357 0.69 MAPT (0.36) MAPTKMT2AMEN1L3MBTL1TDP1
SCHEMBL29520772 0.68 MAPT (0.47) PLK1MAPTKMT2AMEN1HPGD
SCHEMBL18481549 0.67 MAPT (0.46) PLK1MAPTKMT2AMEN1HPGD
SCHEMBL4541307 0.66 CYP19A1 (0.62) MAPTKMT2AMEN1HPGDL3MBTL1
SCHEMBL2730790 0.66 ALDH1A1 (0.50) MAPTKMT2AMEN1HPGDL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002102301-A2 SUBSTITUTED INDOLE-2-CARBOXYLIC ACID BENZYLIDENE-HYDRAZIDES AND ANALOGS AS ACTIVATORS OF CASPASES AND INDUCERS OF APOPTOSIS AND THE USE THEREOF CYTOVIA, INC. (US) 2002-12-27 WO disclosed