SCHEMBL7576846

SCHEMBL7576846

NCc1cccc2nc[nH]c12

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LOXL2 Q9Y4K0 1/20 0.44
PNMT P11086 2/20 0.36
PARP1 P09874 4/20 0.36
PDPK1 O15530 1/20 0.36
CA12 O43570 1/20 0.36
ALOX15 P16050 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
CA9 Q16790 1/20 0.36
TNKS2 Q9H2K2 1/20 0.36
MGMT P16455 1/20 0.35
PIN1 Q13526 1/20 0.35
ASH1L Q9NR48 1/20 0.33
AKT2 P31751 1/20 0.33
HTR3E A5X5Y0 1/20 0.33
MEN1 O00255 1/20 0.33
HTR3B O95264 1/20 0.33
MAPT P10636 1/20 0.33
HTR3A P46098 1/20 0.33
KMT2A Q03164 1/20 0.33
HTR3C Q8WXA8 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3068246 0.85 TAAR1 (0.41) PARP1SMN1; SMN2AKT2MAPT
SCHEMBL2501354 0.81 PARP1 (0.40) PARP1PDPK1CA12ALOX15SMN1; SMN2
SCHEMBL1647059 0.81 PARP1 (0.36) PARP1PDPK1CA12ALOX15SMN1; SMN2
SCHEMBL7346990 0.81 PARP1 (0.43) PARP1PDPK1CA12ALOX15SMN1; SMN2
SCHEMBL30198124 0.79 PARP1 (0.35) PARP1PDPK1CA12ALOX15SMN1; SMN2
SCHEMBL2498957 0.78 MEN1 (0.39) PARP1PDPK1CA12ALOX15SMN1; SMN2
SCHEMBL7856465 0.78 JAK2 (0.36) PARP1PDPK1CA12ALOX15SMN1; SMN2
SCHEMBL20988851 0.77 PARP1 (0.37) PARP1PDPK1CA12ALOX15SMN1; SMN2
SCHEMBL20354325 0.77 GABRA1 (0.44) PARP1PDPK1CA12ALOX15SMN1; SMN2
SCHEMBL21895449 0.75 PARP1 (0.58) LOXL2PARP1PDPK1CA12ALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1250326-A2 INDAZOLE COMPOUNDS, PHARMACEUTICAL COMPOSITIONS, AND THEIR USE FOR MEDIATING OR INHIBITING CELL PROLIFERATION AGOURON PHARMACEUTICALS, INC. (US) 2002-10-23 EP disclosed
WO-2001053268-A2 INDAZOLE COMPOUNDS, PHARMACEUTICAL COMPOSITIONS, AND THEIR USE FOR MEDIATING OR INHIBITING CELL PROLIFERATION AGOURON PHARMACEUTICALS, INC. (US) 2001-07-26 WO disclosed