SCHEMBL7582004

SCHEMBL7582004

CCCOc1cccc(C=O)c1I

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.55
HPGD P15428 1/20 0.55
HTT P42858 1/20 0.55
SMN1; SMN2 Q16637 1/20 0.55
PTGDR2 Q9Y5Y4 1/20 0.42
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42
ERN1 O75460 3/20 0.41
TLR2 O60603 1/20 0.41
TLR1 Q15399 1/20 0.41
TLR6 Q9Y2C9 1/20 0.41
CYP2A6 P11509 1/20 0.41
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
MAPT P10636 1/20 0.39
MCHR1 Q99705 1/20 0.39
SRC P12931 1/20 0.39
AR P10275 1/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8373570 0.86 ALDH1A1 (0.58) ALDH1A1HPGDHTTSMN1; SMN2PTGDR2
SCHEMBL812635 0.84 ALDH1A1 (0.77) ALDH1A1HPGDHTTSMN1; SMN2PTGDR2
SCHEMBL30920025 0.84 ALDH1A1 (0.77) ALDH1A1HPGDHTTSMN1; SMN2PTGDR2
SCHEMBL5724553 0.83 ALDH1A1 (0.58) ALDH1A1HPGDHTTSMN1; SMN2PTGDR2
SCHEMBL29923063 0.83 ALDH1A1 (0.58) ALDH1A1HPGDHTTSMN1; SMN2PTGDR2
SCHEMBL8546246 0.81 ALDH1A1 (0.56) ALDH1A1HPGDHTTSMN1; SMN2PTGDR2
SCHEMBL27659218 0.80 ERN1 (0.62) ALDH1A1HPGDHTTSMN1; SMN2PTGDR2
SCHEMBL15077481 0.80 ALDH1A1 (0.55) ALDH1A1HPGDHTTSMN1; SMN2PTGDR2
SCHEMBL12610716 0.80 ALDH1A1 (0.55) ALDH1A1HPGDHTTSMN1; SMN2PTGDR2
SCHEMBL5030438 0.79 ALDH1A1 (0.48) ALDH1A1HPGDHTTSMN1; SMN2PTGDR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0817782-B1 PHENYL DERIVATIVES USEFUL AS ENDOTHELIN RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM PLC (GB) 2002-09-25 EP disclosed
US-6147111-A KIDNEY, BRAIN, AND CARDIOVASCULAR DISORDERS; VASODILATION SMITHKLINE BEECHAM P.L.C. (GB) 2000-11-14 US disclosed
EP-0817782-A1 PHENYL DERIVATIVES USEFUL AS ENDOTHELIN RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM PLC (GB) 1998-01-14 EP disclosed
WO-1996030358-A1 PHENYL DERIVATIVES USEFUL AS ENDOTHELIN RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM PLC (GB) 1996-10-03 WO disclosed