SCHEMBL7582231

SCHEMBL7582231

COC(=O)C(c1ccc(Cl)nn1)c1ccccc1F

nearest known ligand 0.44

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.44
LMNA P02545 2/20 0.44
ALDH1A1 P00352 3/20 0.38
MEN1 O00255 2/20 0.38
GAA P10253 1/20 0.38
HDAC4 P56524 7/20 0.36
HDAC3 O15379 1/20 0.36
HDAC7 Q8WUI4 1/20 0.36
HDAC8 Q9BY41 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36
HDAC9 Q9UKV0 1/20 0.36
HDAC5 Q9UQL6 1/20 0.36
NCOR2 Q9Y618 1/20 0.36
MC4R P32245 1/20 0.36
CNR2 P34972 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14559834 0.73 ALDH1A1 (0.38) KMT2ALMNAALDH1A1GAA
SCHEMBL13892809 0.71 ALDH1A1 (0.49) KMT2ALMNAALDH1A1GAA
SCHEMBL7116479 0.70 KMT2A (0.47) KMT2ALMNAALDH1A1MEN1GAA
SCHEMBL1274762 0.70 ALDH1A1 (0.56) KMT2ALMNAALDH1A1MEN1GAA
SCHEMBL30059683 0.70 ALDH1A1 (0.56) KMT2ALMNAALDH1A1MEN1GAA
SCHEMBL23879259 0.70 GAA (0.43) KMT2ALMNAALDH1A1GAA
SCHEMBL16111406 0.70 HDAC4 (0.48) KMT2AALDH1A1HDAC4HDAC3HDAC7
SCHEMBL5402848 0.70 GAA (0.50) KMT2ALMNAALDH1A1GAA
SCHEMBL30452188 0.70 GAA (0.43) KMT2ALMNAALDH1A1GAA
SCHEMBL4013185 0.69 MAPK13 (0.39) KMT2AALDH1A1HDAC4HDAC3HDAC7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0810218-B1 6-Benzyl-2H-pyridazin-3-one derivatives,their preparation and their use as inhibitors of prostaglandin G/H synthase I and II (COX I and COX II) HOFFMANN LA ROCHE (CH) 2002-12-04 EP disclosed
US-5886178-A ADMINISTERING OF A PROSTAGLANDIN G/H SYNTHASE INHIBITOR TO A PATIENT TO TREAT INFLAMMATORY OR AUTOIMMUNE DISEASES SYNTEX (U.S.A.) INC. (US) 1999-03-23 US disclosed
EP-0810218-A1 6-Benzyl-2H-pyridazin-3-one derivatives,their preparation and their use as inhibitors of prostaglandin G/H synthase I and II (COX I and COX II) F. HOFFMANN-LA ROCHE AG (CH) 1997-12-03 EP disclosed