SCHEMBL7582908

SCHEMBL7582908

CN(C)CC1=C(c2cccc(O)c2)c2ccccc2C1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 2/20 0.41
CHRM4 P08173 2/20 0.41
CHRM5 P08912 2/20 0.41
CHRM1 P11229 2/20 0.41
CHRM3 P20309 2/20 0.41
HRH1 P35367 2/20 0.41
TSHR P16473 2/20 0.39
KDM4E B2RXH2 1/20 0.39
HSD17B10 Q99714 1/20 0.39
TDP2 O95551 2/20 0.39
ALDH1A1 P00352 1/20 0.37
ATM Q13315 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
ESR1 P03372 1/20 0.36
ESR2 Q92731 1/20 0.36
HSD17B1 P14061 4/20 0.36
HSD17B2 P37059 4/20 0.36
ADRA2A P08913 3/20 0.36
ADRA2B P18089 3/20 0.36
ADRA2C P18825 3/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8017973 0.99 CHRM2 (0.41) CHRM2CHRM4CHRM5CHRM1CHRM3
SCHEMBL7591741 0.89 MTNR1A (0.44) CHRM2CHRM4CHRM5CHRM1CHRM3
Hydrochloric Acid SCHEMBL8010759 0.88 MTNR1A (0.43) CHRM2CHRM4CHRM5CHRM1CHRM3
SCHEMBL7587120 0.87 CHRNB4 (0.40) TSHRKDM4EHSD17B10TDP2ESR1
SCHEMBL7587127 0.87 CHRNB4 (0.40) TSHRKDM4EHSD17B10TDP2ESR1
SCHEMBL7584182 0.87 ESR1 (0.40) TSHRKDM4EHSD17B10TDP2ESR1
Hydrochloric Acid SCHEMBL8011601 0.86 ESR1 (0.39) TSHRKDM4EHSD17B10TDP2ALDH1A1
Hydrochloric Acid SCHEMBL8014791 0.86 CHRNB4 (0.39) TSHRKDM4EHSD17B10TDP2ALDH1A1
Hydrochloric Acid SCHEMBL8014796 0.86 CHRNB4 (0.39) TSHRKDM4EHSD17B10TDP2ALDH1A1
SCHEMBL7588665 0.81 ESR1 (0.40) ESR1ESR2HSD17B1HSD17B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1243721-C Substituted amino compounds and their use as substances having analgesic effect GRUENENTHAL GMBH (DE) 2006-03-01 CN disclosed
EP-0864559-B1 Substituted amino compounds and their use as analgesic active substances GRUENENTHAL GMBH (DE) 2002-06-05 EP disclosed
EP-0864559-A1 Substituted amino compounds and their use as analgesic active substances Grünenthal GmbH (DE) 1998-09-16 EP disclosed