SCHEMBL7585442

SCHEMBL7585442

COc1ccc2c(c1)CCC1(CCN(CC3CC3)CC1)C2=O.Cc1cc(C)c2c(c1)C(=O)C1(CC2)CCN(CC2CC2)CC1

nearest known ligand 0.49

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 6/20 0.49
SIGMAR1 Q99720 4/20 0.49
HTR2A P28223 4/20 0.46
HTR2C P28335 4/20 0.46
HTR2B P41595 2/20 0.46
TNKS O95271 5/20 0.43
TNKS2 Q9H2K2 4/20 0.43
OPRM1 P35372 3/20 0.42
OPRL1 P41146 2/20 0.41
OPRK1 P41145 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
CYP26A1 O43174 1/20 0.37
CYP24A1 Q07973 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6841463 0.89 SIGMAR1 (0.60) DRD2SIGMAR1HTR2AHTR2CHTR2B
SCHEMBL6841136 0.87 SIGMAR1 (0.50) DRD2SIGMAR1HTR2AHTR2CHTR2B
SCHEMBL6841620 0.85 SIGMAR1 (0.64) DRD2SIGMAR1HTR2AHTR2CHTR2B
SCHEMBL6841619 0.84 SIGMAR1 (0.69) DRD2SIGMAR1HTR2AHTR2CHTR2B
SCHEMBL6840788 0.81 SIGMAR1 (0.60) DRD2SIGMAR1HTR2AHTR2CHTR2B
SCHEMBL6840779 0.77 SIGMAR1 (0.64) DRD2SIGMAR1HTR2AHTR2CHTR2B
SCHEMBL6843241 0.76 SIGMAR1 (0.69) DRD2SIGMAR1HTR2AHTR2CHTR2B
SCHEMBL6836319 0.76 SIGMAR1 (0.55) DRD2SIGMAR1HTR2AHTR2CHTR2B
SCHEMBL6841677 0.74 SIGMAR1 (0.62) DRD2SIGMAR1HTR2AHTR2CHTR2B
SCHEMBL6836344 0.74 SIGMAR1 (0.64) DRD2SIGMAR1HTR2AHTR2CHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1235808-A2 TRICYCLIC ANALGESICS WARNER-LAMBERT COMPANY (US) 2002-09-04 EP disclosed
WO-2000075116-A2 TRICYCLIC ANALGESICS WARNER-LAMBERT COMPANY (US) 2000-12-14 WO disclosed