SCHEMBL7586547

SCHEMBL7586547

O=C(NC(=O)c1c(F)cccc1F)Nc1cc(Cl)c(OC(F)(F)C(F)Cl)c(Cl)c1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.57
KMT2A Q03164 3/20 0.57
MAPT P10636 2/20 0.57
USP2 O75604 1/20 0.57
ALOX15 P16050 1/20 0.57
POLB P06746 2/20 0.44
LMNA P02545 1/20 0.44
TLR7 Q9NYK1 3/20 0.44
ATM Q13315 2/20 0.42
NPC1 O15118 2/20 0.41
KDM4E B2RXH2 2/20 0.41
ALDH1A1 P00352 1/20 0.41
MAPK1 P28482 1/20 0.41
PKM P14618 1/20 0.41
RAB9A P51151 1/20 0.41
IL2 P60568 1/20 0.40
TDP1 Q9NUW8 2/20 0.39
TRPA1 O75762 2/20 0.39
GAA P10253 2/20 0.39
THRB P10828 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hexaflumuron SCHEMBL26793 0.93 MEN1 (0.59) MEN1KMT2AMAPTUSP2ALOX15
SCHEMBL10885396 0.92 MEN1 (0.55) MEN1KMT2AMAPTUSP2ALOX15
SCHEMBL7586417 0.91 MEN1 (0.68) MEN1KMT2AMAPTUSP2ALOX15
SCHEMBL7585705 0.90 MEN1 (0.56) MEN1KMT2AMAPTUSP2ALOX15
SCHEMBL9775648 0.89 KMT2A (0.49) MEN1KMT2AMAPTUSP2ALOX15
SCHEMBL7619998 0.89 MEN1 (0.54) MEN1KMT2AMAPTUSP2ALOX15
SCHEMBL10496460 0.88 MEN1 (0.51) MEN1KMT2AMAPTUSP2ALOX15
Hexaflumuron SCHEMBL17607272 0.88 MEN1 (0.53) MEN1KMT2AMAPTUSP2ALOX15
SCHEMBL8659704 0.87 MEN1 (0.63) MEN1KMT2AMAPTUSP2ALOX15
SCHEMBL9804080 0.87 MEN1 (0.52) MEN1KMT2AMAPTUSP2ALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0896532-B1 ACYL UREA COMPOUNDS FOR THE TREATMENT OF COCCIDIOIDOMYCOSIS IN WARM-BLOODED ANIMALS NOVARTIS AG (CH) 2002-10-02 EP claimed
EP-0896532-A1 ACYL UREA COMPOUNDS FOR THE TREATMENT OF COCCIDIOIDOMYCOSIS IN WARM-BLOODED ANIMALS Novartis AG (CH) 1999-02-17 EP claimed
US-5837734-A Method for the treatment of coccidioidomycosis in warm-blooded animals NOVARTIS CORPORATION (US) 1998-11-17 US claimed
WO-1997040826-A1 ACYL UREA COMPOUNDS FOR THE TREATMENT OF COCCIDIOIDOMYCOSIS IN WARM-BLOODED ANIMALS NOVARTIS AG (CH) 1997-11-06 WO claimed
US-5416102-A Administering orally, by injection or implantation, a dosage of flea growth inhibiting benzoyl urea compound CIBA-GEIGY CORPORATION (US) 1995-05-16 US claimed
EP-0896532-B1 ACYL UREA COMPOUNDS FOR THE TREATMENT OF COCCIDIOIDOMYCOSIS IN WARM-BLOODED ANIMALS NOVARTIS AG (CH) 2002-10-02 EP disclosed
EP-0896532-A1 ACYL UREA COMPOUNDS FOR THE TREATMENT OF COCCIDIOIDOMYCOSIS IN WARM-BLOODED ANIMALS Novartis AG (CH) 1999-02-17 EP disclosed
US-5837734-A Method for the treatment of coccidioidomycosis in warm-blooded animals NOVARTIS CORPORATION (US) 1998-11-17 US disclosed
WO-1997040826-A1 ACYL UREA COMPOUNDS FOR THE TREATMENT OF COCCIDIOIDOMYCOSIS IN WARM-BLOODED ANIMALS NOVARTIS AG (CH) 1997-11-06 WO disclosed
US-5416102-A Administering orally, by injection or implantation, a dosage of flea growth inhibiting benzoyl urea compound CIBA-GEIGY CORPORATION (US) 1995-05-16 US disclosed
US-4536341-A INSECTICIDES THE DOW CHEMICAL COMPANY (US) 1985-08-20 US disclosed
US-4468405-A INSECTICIDES THE DOW CHEMICAL COMPANY (US) 1984-08-28 US disclosed