SCHEMBL7586830

SCHEMBL7586830

Cn1c(=O)[nH]cc(C(=O)O)c1=O

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.42
KMT2A Q03164 1/20 0.42
NOTUM Q6P988 1/20 0.42
KDM4E B2RXH2 3/20 0.40
KDM3B Q7LBC6 1/20 0.40
DYRK1A Q13627 1/20 0.36
CSNK2A1 P68400 4/20 0.36
PIM3 Q86V86 1/20 0.36
CLK4 Q9HAZ1 1/20 0.36
CSNK2A2 P19784 3/20 0.35
CSNK2B P67870 3/20 0.35
NAPRT Q6XQN6 1/20 0.34
HPGD P15428 2/20 0.34
CYP2C19 P33261 2/20 0.34
CYP1A2 P05177 1/20 0.34
F7 P08709 1/20 0.33
F3 P13726 1/20 0.33
GAA P10253 1/20 0.33
MAPT P10636 1/20 0.33
HSD17B10 Q99714 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24169816 0.84 PBRM1 (0.39) ALDH1A1KMT2AKDM4EHPGDCYP2C19
SCHEMBL17371768 0.82 ALDH1A1 (0.38) ALDH1A1KDM4EPIM3CYP2C19CYP1A2
SCHEMBL7547639 0.81 KDM3B (0.46) ALDH1A1KMT2ANOTUMKDM4EKDM3B
SCHEMBL22679184 0.79 BRD4 (0.41) ALDH1A1KMT2AKDM4EHPGDCYP2C19
SCHEMBL4284402 0.79 NR4A2 (0.44) ALDH1A1KDM4EHPGDGAA
SCHEMBL19812558 0.78 KDM4E (0.41) ALDH1A1KMT2ANOTUMKDM4EKDM3B
SCHEMBL16863256 0.76 KDM4E (0.41) ALDH1A1KMT2ANOTUMKDM4EKDM3B
SCHEMBL10823654 0.76 PDE4A (0.38) ALDH1A1KMT2ANOTUMKDM4EKDM3B
SCHEMBL6937497 0.75 ALDH1A1 (0.51) ALDH1A1KMT2AKDM4EHPGDCYP2C19
SCHEMBL19243050 0.75 NOTUM (0.40) ALDH1A1KMT2ANOTUMKDM4EKDM3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 35 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-61010565-A None JP disclosed
US-12533354-B2 Triaryl compounds for treatment of PD-L1 diseases CHEMOCENTRYX, INC. (US) 2026-01-27 US disclosed
US-12534450-B2 Methods and compositions for targeting PD-L1 ALIGOS THERAPEUTICS, INC. (US) 2026-01-27 US disclosed
US-20240376078-A1 METHODS AND COMPOSITIONS FOR TARGETING PD-L1 ALIGOS THERAPEUTICS, INC. 2024-11-14 US disclosed
US-20230044941-A1 TRIARYL COMPOUNDS FOR TREATMENT OF PD-L1 DISEASES CHEMOCENTRYX, INC. 2023-02-09 US disclosed
US-20230044941-A1 TRIARYL COMPOUNDS FOR TREATMENT OF PD-L1 DISEASES CHEMOCENTRYX, INC. 2023-02-09 US disclosed
US-20230031213-A1 METHODS AND COMPOSITIONS FOR TARGETING PD-L1 ALIGOS THERAPEUTICS, INC. 2023-02-02 US disclosed
CN-114340633-A Triaryl compounds for the treatment of PD-L1 disease 凯莫森特里克斯股份有限公司 2022-04-12 CN disclosed
EP-3968996-A1 TRIARYL COMPOUNDS FOR TREATMENT OF PD-L1 DISEASES ChemoCentryx, Inc. (US) 2022-03-23 EP disclosed
US-11266643-B2 Triaryl compounds for treatment of PD-L1 diseases CHEMOCENTRYX, INC. (US) 2022-03-08 US disclosed
WO-1996017832-A1 NOVEL GLUTAMATE RECEPTOR ANTAGONISTS: FUSED CYCLOALKYLQUINOXALINEDIONES WARNER-LAMBERT COMPANY (US) 1996-06-13 WO disclosed
EP-0649443-A4 OXAZOLONE DERIVED MATERIALS. LEGOMER PARTNERS LP (US) 1995-11-08 EP disclosed
WO-1995018186-A1 MODULAR DESIGN AND SYNTHESIS OF AMINIMIDE CONTAINING MOLECULES ARQULE PARTNERS, L.P. (US) 1995-07-06 WO disclosed
WO-1995017903-A1 MODULAR DESIGN AND SYNTHESIS OF OXAZOLONE-DERIVED MOLECULES ARQULE PARTNERS, L.P. (US) 1995-07-06 WO disclosed
EP-0649443-A1 OXAZOLONE DERIVED MATERIALS LEGOMER PARTNERS, L.P. (US) 1995-04-26 EP disclosed
WO-1994000509-A9 OXAZOLONE DERIVED MATERIALS 1994-03-17 WO disclosed
WO-1994001102-A1 AMINIMIDE-CONTAINING MOLECULES AND MATERIALS AS MOLECULAR RECOGNITION AGENTS LEGOMER PARTNERS, L.P. (US) 1994-01-20 WO disclosed
WO-1994000509-A1 OXAZOLONE DERIVED MATERIALS LEGOMER PARTNERS, L.P. (US) 1994-01-06 WO disclosed
JP-S6110565-A PREPARATION OF URACIL-5-CARBOXYLIC ACID ESTER TAKEDA CHEM IND LTD 1986-01-18 JP disclosed
US-3953428-A ANTIBACTERIAL YAMANOUCHI PHARMACEUTICAL CO., LTD. (JA) 1976-04-27 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12533354-B2 Triaryl compounds for treatment of PD-L1 diseases CD274, PDCD1LG2, PDCD1 ALDH1A1 388/4885KMT2A 1574/4885NOTUM 4629/4885
US-12534450-B2 Methods and compositions for targeting PD-L1 CD274, PDCD1LG2, PDCD1 ALDH1A1 608/4885KMT2A 2186/4885NOTUM 4807/4885
US-20230031213-A1 METHODS AND COMPOSITIONS FOR TARGETING PD-L1 CD274, PDCD1LG2, PDCD1 ALDH1A1 301/4885KMT2A 2794/4885NOTUM 4082/4885
US-20230044941-A1 TRIARYL COMPOUNDS FOR TREATMENT OF PD-L1 DISEASES CD274, PDCD1, PDCD1LG2 ALDH1A1 380/4885KMT2A 568/4885NOTUM 4282/4885
US-20240376078-A1 METHODS AND COMPOSITIONS FOR TARGETING PD-L1 CD274, PDCD1LG2, PDCD1 ALDH1A1 301/4885KMT2A 2794/4885NOTUM 4082/4885
US-11266643-B2 Triaryl compounds for treatment of PD-L1 diseases CD274, PDCD1, PDCD1LG2 ALDH1A1 380/4885KMT2A 568/4885NOTUM 4282/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.