SCHEMBL7587498

SCHEMBL7587498

C[SiH](C)Oc1ccc(C(C)(C)CBr)cc1

nearest known ligand 0.37

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.37
MAPT P10636 1/20 0.37
RAB9A P51151 1/20 0.37
SMN1; SMN2 Q16637 2/20 0.35
CYP3A4 P08684 1/20 0.35
APP P05067 1/20 0.32
SHBG P04278 1/20 0.31
MAOB P27338 1/20 0.30
HRH3 Q9Y5N1 1/20 0.30
ACACB O00763 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7178856 0.78 SHBG (0.42) NPC1MAPTRAB9ASMN1; SMN2CYP3A4
SCHEMBL7904973 0.78 SMN1; SMN2 (0.44) NPC1MAPTRAB9ASMN1; SMN2CYP3A4
SCHEMBL30407868 0.73 CA1 (0.39)
SCHEMBL11503011 0.72 TSHR (0.48) NPC1MAPTRAB9AAPPSHBG
SCHEMBL15029224 0.71 CA1 (0.44) NPC1MAPTRAB9ASMN1; SMN2CYP3A4
SCHEMBL17961713 0.70 TSHR (0.52) NPC1MAPTRAB9ASHBG
SCHEMBL14828478 0.69 ESR2 (0.61) MAPTCYP3A4SHBG
SCHEMBL2497844 0.69 SHBG (0.61) CYP3A4SHBG
SCHEMBL22366368 0.68 APP (0.39) CYP3A4APP
SCHEMBL10953696 0.68 CYP2A6 (0.42) NPC1MAPTRAB9AAPPMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0944613-B1 BENZOPYRAN DERIVATIVES CHUGAI PHARMACEUTICAL CO LTD (JP) 2002-10-09 EP disclosed
US-6153768-A RECEPTOR BLOCKING ANTIESTROGENS HAVING REDUCED SIDE EFFECTS C & C RESEARCH LABORATORIES (KR) 2000-11-28 US disclosed
US-5561143-A ANTICHOLESTEROL AGENTS, ANTILIPEMIC AGENTS RHONE-POULENC RORER PHARMACEUTICALS INC. (US) 1996-10-01 US disclosed
US-5534532-A ANTICHOLESTEROL AGENTS, SQUALENE SYNTHASE INHIBITOR RHONE-POULENC RORER PHARMACEUTICALS INC. (US) 1996-07-09 US disclosed
US-5455260-A Anticholesterol agents; reduction of serum cholesterol without reducing mevalonic metabolite synthesis; side effect RHONE-POULENC RORER PHARMACEUTICALS INC. (US) 1995-10-03 US disclosed
WO-1994027601-A1 ALIPHATIC AMINO BIS-ARYL SQUALENE SYNTHASE INHIBITORS RHONE-POULENC RORER PHARMACEUTICALS INC. (US) 1994-12-08 WO disclosed