SCHEMBL7590367

SCHEMBL7590367

CCc1nc2c(-c3c(C)cc(C)cc3C)cccc2n1C(CC)CC

nearest known ligand 0.43

Predicted protein targets (top 1)

geneUniProtsupporting neighboursconfidence
CRHR1 P34998 6/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7813333 0.78
SCHEMBL8006443 0.75 CRHR1 (0.40) CRHR1
SCHEMBL6839583 0.74 CRHR1 (0.30) CRHR1
SCHEMBL7806586 0.74 CRHR1 (0.38) CRHR1
SCHEMBL22833928 0.73 CRHR1 (0.38) CRHR1
SCHEMBL29501666 0.73 CRHR1 (0.38) CRHR1
SCHEMBL7806584 0.72 CRHR1 (0.38) CRHR1
SCHEMBL29873429 0.72 KMT2A (0.38) CRHR1
SCHEMBL22855416 0.72 KMT2A (0.38) CRHR1
SCHEMBL22855428 0.70 CRHR1 (0.41) CRHR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0812831-B1 Benzimidazole derivatives and their use as corticotropin releasing factor antagonists PFIZER (US) 2002-09-04 EP disclosed
US-6022978-A Benzimidazole derivatives PFIZER INC. (US) 2000-02-08 US disclosed
EP-0812831-A1 Benzimidazole derivatives and their use as corticotropin releasing factor antagonists PFIZER INC. (US) 1997-12-17 EP disclosed