SCHEMBL7591539

SCHEMBL7591539

CC(NC1CCc2[nH]c3ccccc3c2C1)c1ccccc1

nearest known ligand 0.60

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NR2E1 Q9Y466 1/20 0.53
GAA P10253 1/20 0.49
L3MBTL1 Q9Y468 1/20 0.49
RB1 P06400 5/20 0.48
TP53 P04637 1/20 0.44
HPGD P15428 1/20 0.44
HSD17B10 Q99714 1/20 0.44
CYP2D6 P10635 1/20 0.44
KCNH2 Q12809 1/20 0.44
HTR1A P08908 1/20 0.42
HTR1D P28221 1/20 0.42
HTR1B P28222 1/20 0.42
HTR2A P28223 1/20 0.41
HTR2C P28335 1/20 0.41
AHR P35869 1/20 0.41
DRD2 P14416 1/20 0.41
DRD1 P21728 1/20 0.41
DRD5 P21918 1/20 0.41
SLC2A1 P11166 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9834959 1.00 NR2E1 (0.53) NR2E1GAAL3MBTL1RB1TP53
SCHEMBL7591546 1.00 NR2E1 (0.53) NR2E1GAAL3MBTL1RB1TP53
Sulfuric Acid SCHEMBL7589746 0.93 NR2E1 (0.47) NR2E1GAAL3MBTL1RB1TP53
SCHEMBL14768417 0.86 VPS4B (0.51) GAAL3MBTL1CYP2D6KCNH2HTR1A
SCHEMBL2494316 0.86 VPS4B (0.51) GAAL3MBTL1CYP2D6KCNH2HTR1A
SCHEMBL2494312 0.86 VPS4B (0.51) GAAL3MBTL1CYP2D6KCNH2HTR1A
SCHEMBL2493068 0.86 VPS4B (0.51) GAAL3MBTL1CYP2D6KCNH2HTR1A
SCHEMBL2493069 0.86 VPS4B (0.51) GAAL3MBTL1CYP2D6KCNH2HTR1A
SCHEMBL4803895 0.81 NR2E1 (0.61) NR2E1GAARB1TP53HPGD
SCHEMBL23875579 0.79 NR2E1 (0.58) NR2E1RB1TP53HPGDHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010078250-A1 SYNTHESIS OF (2-AMINO)-TETRAHYDROCARBAZOLE-PROPANOIC ACID CHIRAL QUEST, INC. (US) 2010-07-08 WO disclosed
EP-0728743-B1 3-Amino-tetrahydrocarbazol propanoic acid esters BAYER AG (DE) 2002-10-30 EP disclosed
US-5684158-A 3-amino!-tetrahydrocarbazole-propanoic acid esters BAYER AKTIENGESELLSCHAFT (DE) 1997-11-04 US disclosed
EP-0728743-A1 3-Amino-tetrahydrocarbazol propanoic acid esters BAYER AG (DE) 1996-08-28 EP disclosed