SCHEMBL7592018

SCHEMBL7592018

CCc1ccc(CC(=O)N(C)C)cc1N

nearest known ligand 0.43

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.43
ALDH1A1 P00352 1/20 0.41
GAA P10253 1/20 0.41
GFER P55789 1/20 0.41
NUDT1 P36639 1/20 0.41
CHEK1 O14757 2/20 0.40
PCNA P12004 1/20 0.37
HDAC4 P56524 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36
POLB P06746 1/20 0.36
APEX1 P27695 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
SLC6A2 P23975 1/20 0.35
SLC6A4 P31645 1/20 0.35
BACE1 P56817 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19182412 0.88 PARP1 (0.43) PARP1ALDH1A1GAAGFERNUDT1
SCHEMBL10665217 0.86 PARP1 (0.46) PARP1ALDH1A1GAAGFERNUDT1
SCHEMBL10175368 0.83 PARP1 (0.43) PARP1NUDT1PCNAHDAC4HDAC6
SCHEMBL28229854 0.80 PARP1 (0.42) PARP1ALDH1A1GAAGFERNUDT1
SCHEMBL5094928 0.79 GAA (0.53) PARP1ALDH1A1GAAGFERNUDT1
SCHEMBL19180433 0.79 SKP2 (0.46) PARP1ALDH1A1GAAGFERNUDT1
SCHEMBL18772546 0.79 PRKCI (0.49) PARP1ALDH1A1GAAGFERNUDT1
SCHEMBL19181011 0.78 PARP1 (0.43) PARP1ALDH1A1GAAGFERNUDT1
SCHEMBL5100488 0.78 ALDH1A1 (0.51) ALDH1A1GAAGFERCHEK1
SCHEMBL19180323 0.78 CYP3A4 (0.52) PARP1NUDT1CHEK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6368573-B1 MEASURING MYOCARDIAL FUNCTION IN MAMMAL KING PHARMACEUTICALS RESEARCH AND DEVELOPMENT, INC. 2002-04-09 US disclosed
US-5063233-A Cardiovascular disorders CIBA-GEIGY CORPORATION (US) 1991-11-05 US disclosed
US-5034381-A Antagonist CIBA-GEIGY CORPORATION (US) 1991-07-23 US disclosed
US-4968697-A ADENOSINE-2 RECEPTOR AGONISTS CIBA-GEIGY CORPORATION (US) 1990-11-06 US disclosed
US-4954504-A Hypotensive agents, psychotic disorders CIBA-GEIGY CORPORATION (US) 1990-09-04 US disclosed
EP-0323807-A2 Certain 2-substituted adenosine derivatives CIBA-GEIGY AG (CH) 1989-07-12 EP disclosed
EP-0277917-A2 Certain adenosine 5'-carboxamide derivatives CIBA-GEIGY AG (CH) 1988-08-10 EP disclosed
EP-0267878-A1 N9-cyclopentyl-substituted adenine derivatives CIBA-GEIGY AG (CH) 1988-05-18 EP disclosed