SCHEMBL7597158

SCHEMBL7597158

O=C(NC(=S)Nc1ccc(CCN(Cc2cccc(Cl)c2)C(=O)C(F)(F)F)cc1)c1ccccc1

nearest known ligand 0.55

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.50
NPSR1 Q6W5P4 2/20 0.50
NPC1 O15118 1/20 0.50
EPHX1 P07099 1/20 0.50
RAB9A P51151 1/20 0.50
KCNH2 Q12809 1/20 0.48
SMN1; SMN2 Q16637 2/20 0.47
MAPT P10636 1/20 0.47
POLB P06746 1/20 0.47
CYP2C9 P11712 1/20 0.45
ALOX12 P18054 1/20 0.45
CYP2C19 P33261 1/20 0.45
HTT P42858 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7599280 0.76 LPAR1 (0.43) ALDH1A1KCNH2
SCHEMBL7597734 0.73 POLB (0.59) ALDH1A1NPSR1NPC1EPHX1RAB9A
SCHEMBL7598234 0.73 KCNH2 (0.57) ALDH1A1NPC1RAB9AKCNH2SMN1; SMN2
SCHEMBL3059584 0.72 SMN1; SMN2 (0.69) ALDH1A1NPSR1NPC1EPHX1RAB9A
SCHEMBL3049551 0.71 NPC1 (0.78) ALDH1A1NPSR1NPC1EPHX1RAB9A
SCHEMBL7597743 0.70 POLB (0.67) ALDH1A1NPSR1NPC1EPHX1RAB9A
SCHEMBL3055302 0.70 SMN1; SMN2 (0.69) ALDH1A1NPC1RAB9ASMN1; SMN2MAPT
SCHEMBL3050273 0.69 ALDH1A1 (0.68) ALDH1A1NPSR1NPC1EPHX1RAB9A
SCHEMBL3059631 0.69 ALDH1A1 (0.76) ALDH1A1NPSR1NPC1EPHX1RAB9A
SCHEMBL8611590 0.69 ALDH1A1 (0.84) ALDH1A1NPSR1NPC1EPHX1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0782567-B2 ISOTHIOUREA DERIVATIVES AS NO SYNTHASE INHIBITORS ASTRA AB (SE) 2002-12-11 EP disclosed
EP-0782567-B1 ISOTHIOUREA DERIVATIVES AS NO SYNTHASE INHIBITORS ASTRA AB (SE) 1999-06-30 EP disclosed
US-5721247-A Isothiourea derivatives useful in therapy ASTRA AKTIEBOLAG (SE) 1998-02-24 US disclosed