SCHEMBL7599286

SCHEMBL7599286

COc1ccc(C2(C#Cc3ccncc3)CCC3(CC2)OCCO3)cc1OC1CCCC1

nearest known ligand 0.49

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 19/20 0.49
PDE4B Q07343 18/20 0.49
PDE4C Q08493 18/20 0.49
PDE4D Q08499 18/20 0.49
S1PR1 P21453 1/20 0.43
S1PR3 Q99500 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7419473 0.88 PDE4A (0.53) PDE4APDE4BPDE4CPDE4D
SCHEMBL6172676 0.85 PDE4A (0.52) PDE4APDE4BPDE4CPDE4D
SCHEMBL6172674 0.85 PDE4A (0.52) PDE4APDE4BPDE4CPDE4D
SCHEMBL8508309 0.85 PDE4A (0.46) PDE4APDE4BPDE4CPDE4D
SCHEMBL7408401 0.85 PDE4A (0.47) PDE4APDE4BPDE4CPDE4D
SCHEMBL8511338 0.85 PDE4A (0.49) PDE4APDE4BPDE4CPDE4D
SCHEMBL7375913 0.85 PDE4A (0.68) PDE4APDE4BPDE4CPDE4D
SCHEMBL7404582 0.84 PDE4A (0.46) PDE4APDE4BPDE4CPDE4D
SCHEMBL8510180 0.84 PDE4A (0.44) PDE4APDE4BPDE4CPDE4D
SCHEMBL8357454 0.83 PDE4A (0.51) PDE4APDE4BPDE4CPDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5861421-A 4,4-(disubstituted) cyclohexan-1-one monomers and related compounds SMITHKLINE BEECHAM CORPORATION (US) 1999-01-19 US disclosed
EP-0800393-A4 4,4-(DISUBSTITUTED)CYCLOHEXAN-1-ONE MONOMERS AND RELATED COMPOUNDS SMITHKLINE BEECHAM CORP (US) 1998-05-06 EP disclosed
EP-0800393-A1 4,4-(DISUBSTITUTED)CYCLOHEXAN-1-ONE MONOMERS AND RELATED COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 1997-10-15 EP disclosed
WO-1996019995-A1 4,4-(DISUBSTITUTED)CYCLOHEXAN-1-ONE MONOMERS AND RELATED COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 1996-07-04 WO disclosed